BDBM185699 UNC10108049::US9156822, 43

SMILES CC(=O)Nc1cc(OCCCCN2CCN(CC2)c2cccc(Cl)c2Cl)ccc1C

InChI Key InChIKey=PYODBBFAXCRGHN-UHFFFAOYSA-N

Data  1 KI  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 185699   

TargetD(2) dopamine receptor(Human)
University of North Carolina at Chapel Hill

US Patent
LigandPNGBDBM185699(UNC10108049 | US9156822, 43)
Affinity DataEC50:  9.20nMpH: 7.4Assay Description:Recruitment of β-arrestin to agonist-stimulated D2 receptors was performed using a previously described Tango-type assay (Barnea et al., Proc. N...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2016
Entry Details
US Patent

TargetD(2) dopamine receptor(Human)
University of North Carolina at Chapel Hill

US Patent
LigandPNGBDBM185699(UNC10108049 | US9156822, 43)
Affinity DataKi:  72nMpH: 7.4Assay Description:Membranes prepared as above were resuspended to 1 ug protein/ul (measured by Bradford assay using BSA as standard), and 50 ul were added to each well...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2016
Entry Details
US Patent