BDBM18613 6-bisalkylamino-2-quinolinone, 8d::6-{[(2S)-1-chloropropan-2-yl](2,2,2-trifluoroethyl)amino}-4-(trifluoromethyl)-1,2-dihydroquinolin-2-one

SMILES C[C@@H](CCl)N(CC(F)(F)F)c1ccc2[nH]c(=O)cc(c2c1)C(F)(F)F

InChI Key InChIKey=AUIQVMLZIOYPBH-QMMMGPOBSA-N

Data  1 KI  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 18613   

TargetAndrogen receptor(Homo sapiens (Human))
Ligand Pharmaceuticals

LigandPNGBDBM18613(6-bisalkylamino-2-quinolinone, 8d | 6-{[(2S)-1-chl...)
Affinity DataKi:  9.80nM EC50:  3.60nMAssay Description:The compounds were evaluated in a transcriptional activation assay with hAR in a mammalian cell background (CV-1) as the primary in vitro assay. Rece...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed