BDBM186573 US10787472, Compound 9::US20230303497, Example VX-150::US9163042, 9
SMILES: Cc1cc(F)ccc1Oc1cc(ccc1C(=O)Nc1ccn(COP(O)(O)=O)c(=O)c1)C(F)(F)F
InChI Key: InChIKey=SQDQNNKQTHOQHO-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 5 hits for monomerid = 186573 Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
Sodium channel protein type 10 subunit alpha
(Rat) | BDBM186573
 (US9163042, 9 | US10787472, Compound 9 | US20230303...) | GoogleScholar
| UniChem
| | n/a | n/a | 330 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this Ligand-Target Pair | |
Sodium channel protein type 10 subunit alpha
(Human) | BDBM186573
 (US9163042, 9 | US10787472, Compound 9 | US20230303...) | GoogleScholar
| UniChem
| | n/a | n/a | 330 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this Ligand-Target Pair | |
Potassium voltage-gated channel subfamily H member 2
(Human) | BDBM186573
 (US9163042, 9 | US10787472, Compound 9 | US20230303...) | GoogleScholar
| UniChem
| | n/a | n/a | 7.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this Ligand-Target Pair | |
Sodium channel protein type 10 subunit alpha
(Human) | BDBM186573
 (US9163042, 9 | US10787472, Compound 9 | US20230303...) | GoogleScholar
| UniChem
| | n/a | n/a | 33 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this Ligand-Target Pair | |
Sodium channel protein type 10 subunit alpha
(Human) | BDBM186573
 (US9163042, 9 | US10787472, Compound 9 | US20230303...) | GoogleScholar
| UniChem
| | n/a | n/a | 86 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this Ligand-Target Pair | |