BDBM198063 US9221795, 59

SMILES Nc1nc(N)c(Cl)c(N[C@@H](C2CC2)c2nc3c(F)ccc(C#N)c3c(=O)n2-c2cccnc2)n1

InChI Key InChIKey=NHZVHHAMKTUMFU-INIZCTEOSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 198063   

TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Gilead Sciences

US Patent
LigandPNGBDBM198063(US9221795, 59)
Affinity DataIC50:  380nMpH: 7.4Assay Description:Class I PI3K isoforms were expressed and purified as heterodimeric recombinant proteins. All assay reagents and buffers for the TR-FRET assay were pu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent