BDBM20028 (5Z)-5-({4-[({3-[3-benzoyl-8-(trifluoromethyl)quinolin-4-yl]phenyl}amino)methyl]phenyl}methylidene)-1,3-thiazolidine-2,4-dione::(5Z)-5-{4-[({3-[3-Benzoyl-8-(trifluoromethyl)quinolin-4-yl]phenyl} amino)methyl] benzylidene}-1,3-thiazolidine-2,4-dione::thiazolidine-2,4-dione, 40

SMILES FC(F)(F)c1cccc2c(-c3cccc(NCc4ccc(\C=C5/SC(=O)NC5=O)cc4)c3)c(cnc12)C(=O)c1ccccc1

InChI Key InChIKey=JPIHSYRXQLKCID-NTFVMDSBSA-N

Data  2 IC50  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 20028   

TargetOxysterols receptor LXR-beta [154-461](Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM20028((5Z)-5-({4-[({3-[3-benzoyl-8-(trifluoromethyl)quin...)
Affinity DataIC50:  276nM EC50:  369nMAssay Description:Binding reaction was initiated by adding a dilution series of test compound in tracer solution to LXR-coated flash plates. Each concentration of test...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha [197-447](Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM20028((5Z)-5-({4-[({3-[3-benzoyl-8-(trifluoromethyl)quin...)
Affinity DataIC50:  456nMpH: 7.4 T: 2°CAssay Description:Binding reaction was initiated by adding a dilution series of test compound in tracer solution to LXR-coated flash plates. Each concentration of test...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed