BDBM200372 US10011599, Example 1A::US9227969, 1A::US9629836, 1A
SMILES: Cc1nc2cnc3cc(F)c(cc3c2n1[C@H]1CCN(C[C@@H]1F)C(=O)CO)-c1ccc(Oc2ncccn2)cc1Cl
InChI Key: InChIKey=WZZBNLYBHUDSHF-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 5 hits for monomerid = 200372 Target/Host
(Institution) | Ligand | Target/Host
Links | Ligand
Links | Trg + Lig
Links | Ki
nM | ΔG°
kcal/mole | IC50
nM | Kd
nM | EC50
nM | koff
s-1 | kon
M-1s-1 | pH | Temp
°C |
|---|
Dual specificity mitogen-activated protein kinase kinase 1 [K97R]
(Human) | BDBM200372
(US9227969, 1A | US9629836, 1A | US10011599, Exampl...) | GoogleScholar
| UniChem
| | n/a | n/a | 5 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Dual specificity mitogen-activated protein kinase kinase 1
(Human) | BDBM200372
(US9227969, 1A | US9629836, 1A | US10011599, Exampl...) | GoogleScholar
| UniChem
| | n/a | n/a | 5 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Dual specificity mitogen-activated protein kinase kinase 1/Mitogen-activated protein kinase 1/Serine/threonine-protein kinase B-raf
(Human) | BDBM200372
(US9227969, 1A | US9629836, 1A | US10011599, Exampl...) | GoogleScholar
| UniChem
| | n/a | n/a | 5 | n/a | n/a | n/a | n/a | 7.5 | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
Cytochrome P450 3A4
(Human) | BDBM200372
(US9227969, 1A | US9629836, 1A | US10011599, Exampl...) | GoogleScholar
| UniChem
| | n/a | n/a | 7.70E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
High affinity nerve growth factor receptor
(Human) | BDBM200372
(US9227969, 1A | US9629836, 1A | US10011599, Exampl...) | GoogleScholar
| UniChem
| | n/a | n/a | 25 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
|
More data for this
Ligand-Target Pair | |
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