BDBM20434 1-[(4-bromophenyl)methyl]-3-1H-indazol-5-ylurea::heterocyclic urea, 33

SMILES Brc1ccc(CNC(=O)Nc2ccc3[nH]ncc3c2)cc1

InChI Key InChIKey=NPLQZQGAZAUUTB-UHFFFAOYSA-N

Data  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 20434   

TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Abbott Laboratories

LigandPNGBDBM20434(1-[(4-bromophenyl)methyl]-3-1H-indazol-5-ylurea | ...)
Affinity DataEC50:  3.54E+3nMpH: 7.4 T: 2°CAssay Description:The functional antagonist activity of compounds at the TRPV1 receptor was determined with a Ca2+ influx assay by measuring the effect on capsaicin (0...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed