BDBM20461 (6E)-N-[(4-hydroxy-3-methoxyphenyl)methyl]-8-methylnon-6-enamide::(E)-N-[(4-hydroxy-3-methoxyphenyl)methyl]-8-methylnon-6-enamide::CAP::CHEMBL294199::Capsaicin::Zostrix

SMILES: CC(C)/C=C/CCCCC(=O)NCc1ccc(c(c1)OC)O

InChI Key: InChIKey=YKPUWZUDDOIDPM-UHFFFAOYSA-N

Data: 15 KI  18 IC50  27 EC50

PDB links: 7 PDB IDs match this monomer.

Find this compound or compounds like it in BindingDB or PDB:

Substructure Similarity at least:  must be >=0.5 Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 59 hits for monomerid = 20461   

Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50 nM	koff s-1	kon M-1s-1	pH	Temp °C
Prostaglandin G/H synthase 1 (Human)	BDBM20461 (Zostrix | (E)-N-[(4-hydroxy-3-methoxyphenyl)methyl...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	3.80E+3	n/a	n/a	n/a	n/a	n/a	n/a
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Transient receptor potential cation channel subfamily V member 1 (Human)	BDBM20461 (Zostrix | (E)-N-[(4-hydroxy-3-methoxyphenyl)methyl...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	n/a	45	n/a	n/a	n/a	n/a
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Lysine-specific histone demethylase 1A (Human)	BDBM20461 (Zostrix | (E)-N-[(4-hydroxy-3-methoxyphenyl)methyl...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	600	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
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Lysine-specific histone demethylase 1A (Human)	BDBM20461 (Zostrix | (E)-N-[(4-hydroxy-3-methoxyphenyl)methyl...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	600	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily V member 1 (Human)	BDBM20461 (Zostrix | (E)-N-[(4-hydroxy-3-methoxyphenyl)methyl...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	n/a	29	n/a	n/a	n/a	n/a
TBA									Citation and Details
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Lysine-specific histone demethylase 1A (Human)	BDBM20461 (Zostrix | (E)-N-[(4-hydroxy-3-methoxyphenyl)methyl...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	600	n/a	n/a	n/a	n/a	n/a	n/a
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Transient receptor potential cation channel subfamily M member 8 (Human)	BDBM20461 (Zostrix | (E)-N-[(4-hydroxy-3-methoxyphenyl)methyl...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	1.00E+3	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily V member 1 (Human)	BDBM20461 (Zostrix | (E)-N-[(4-hydroxy-3-methoxyphenyl)methyl...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	n/a	5	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily V member 1 (Human)	BDBM20461 (Zostrix | (E)-N-[(4-hydroxy-3-methoxyphenyl)methyl...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	8	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily V member 1 (Human)	BDBM20461 (Zostrix | (E)-N-[(4-hydroxy-3-methoxyphenyl)methyl...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	420	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily V member 1 (Human)	BDBM20461 (Zostrix | (E)-N-[(4-hydroxy-3-methoxyphenyl)methyl...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	313	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily V member 1 (Rat)	BDBM20461 (Zostrix | (E)-N-[(4-hydroxy-3-methoxyphenyl)methyl...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	19	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily V member 1 (Human)	BDBM20461 (Zostrix | (E)-N-[(4-hydroxy-3-methoxyphenyl)methyl...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	n/a	3.90	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily V member 1 (Human)	BDBM20461 (Zostrix | (E)-N-[(4-hydroxy-3-methoxyphenyl)methyl...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	n/a	40	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Lysine-specific histone demethylase 1A (Human)	BDBM20461 (Zostrix | (E)-N-[(4-hydroxy-3-methoxyphenyl)methyl...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	600	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily V member 1 (Rat)	BDBM20461 (Zostrix | (E)-N-[(4-hydroxy-3-methoxyphenyl)methyl...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	n/a	44.8	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily V member 1 (Human)	BDBM20461 (Zostrix | (E)-N-[(4-hydroxy-3-methoxyphenyl)methyl...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	n/a	40	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily V member 1 (Human)	BDBM20461 (Zostrix | (E)-N-[(4-hydroxy-3-methoxyphenyl)methyl...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	n/a	2.51	n/a	n/a	n/a	n/a
TBA									Citation and Details
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Transient receptor potential cation channel subfamily M member 8 (Mouse)	BDBM20461 (Zostrix | (E)-N-[(4-hydroxy-3-methoxyphenyl)methyl...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	>1.00E+5	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily M member 8 (Mouse)	BDBM20461 (Zostrix | (E)-N-[(4-hydroxy-3-methoxyphenyl)methyl...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	2.80E+4	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily V member 1 (Human)	BDBM20461 (Zostrix | (E)-N-[(4-hydroxy-3-methoxyphenyl)methyl...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	8	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily V member 1 (Human)	BDBM20461 (Zostrix | (E)-N-[(4-hydroxy-3-methoxyphenyl)methyl...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	n/a	5.30	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily V member 1/2/4 (Rat)	BDBM20461 (Zostrix | (E)-N-[(4-hydroxy-3-methoxyphenyl)methyl...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	n/a	30	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily V member 1/2/4 (Rat)	BDBM20461 (Zostrix | (E)-N-[(4-hydroxy-3-methoxyphenyl)methyl...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	n/a	300	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily V member 1/2/4 (Rat)	BDBM20461 (Zostrix | (E)-N-[(4-hydroxy-3-methoxyphenyl)methyl...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	n/a	300	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily V member 1/2/4 (Rat)	BDBM20461 (Zostrix | (E)-N-[(4-hydroxy-3-methoxyphenyl)methyl...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	n/a	300	n/a	n/a	n/a	n/a
TBA									Citation and Details
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Potassium voltage-gated channel subfamily A member 1 (Human)	BDBM20461 (Zostrix | (E)-N-[(4-hydroxy-3-methoxyphenyl)methyl...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	2.90E+4	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily V member 1 (Rat)	BDBM20461 (Zostrix | (E)-N-[(4-hydroxy-3-methoxyphenyl)methyl...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	n/a	45	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily V member 1 (Human)	BDBM20461 (Zostrix | (E)-N-[(4-hydroxy-3-methoxyphenyl)methyl...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	n/a	870	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily V member 1 (Human)	BDBM20461 (Zostrix | (E)-N-[(4-hydroxy-3-methoxyphenyl)methyl...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	n/a	1.00E+3	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily V member 1/2/4 (Rat)	BDBM20461 (Zostrix | (E)-N-[(4-hydroxy-3-methoxyphenyl)methyl...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	n/a	300	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily V member 1 (Human)	BDBM20461 (Zostrix | (E)-N-[(4-hydroxy-3-methoxyphenyl)methyl...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	n/a	20	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily V member 1 (Rat)	BDBM20461 (Zostrix | (E)-N-[(4-hydroxy-3-methoxyphenyl)methyl...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	n/a	2.32E+3	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily V member 1 (Rat)	BDBM20461 (Zostrix | (E)-N-[(4-hydroxy-3-methoxyphenyl)methyl...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	n/a	44.8	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily V member 1 (Human)	BDBM20461 (Zostrix | (E)-N-[(4-hydroxy-3-methoxyphenyl)methyl...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	n/a	871	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily V member 1 (Human)	BDBM20461 (Zostrix | (E)-N-[(4-hydroxy-3-methoxyphenyl)methyl...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	n/a	26	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily V member 1 (Human)	BDBM20461 (Zostrix | (E)-N-[(4-hydroxy-3-methoxyphenyl)methyl...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	n/a	7.20	n/a	n/a	n/a	n/a
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Polyunsaturated fatty acid 5-lipoxygenase (Human)	BDBM20461 (Zostrix | (E)-N-[(4-hydroxy-3-methoxyphenyl)methyl...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	5.60E+4	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily V member 1 (Human)	BDBM20461 (Zostrix | (E)-N-[(4-hydroxy-3-methoxyphenyl)methyl...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	n/a	5.30	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily V member 1 (Human)	BDBM20461 (Zostrix | (E)-N-[(4-hydroxy-3-methoxyphenyl)methyl...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	8	n/a	n/a	n/a	n/a	n/a	n/a
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Acetylcholinesterase (Human)	BDBM20461 (Zostrix | (E)-N-[(4-hydroxy-3-methoxyphenyl)methyl...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	>2.00E+5	n/a	n/a	n/a	n/a	n/a	n/a
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Bile salt export pump (Human)	BDBM20461 (Zostrix | (E)-N-[(4-hydroxy-3-methoxyphenyl)methyl...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	<1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily V member 1 (Human)	BDBM20461 (Zostrix | (E)-N-[(4-hydroxy-3-methoxyphenyl)methyl...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	n/a	3.02E+4	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily V member 1 (Human)	BDBM20461 (Zostrix | (E)-N-[(4-hydroxy-3-methoxyphenyl)methyl...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	n/a	20	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily V member 1 (Human)	BDBM20461 (Zostrix | (E)-N-[(4-hydroxy-3-methoxyphenyl)methyl...) Show SMILES Show InChI	GoogleScholar	UniChem		6	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily V member 1 (Human)	BDBM20461 (Zostrix | (E)-N-[(4-hydroxy-3-methoxyphenyl)methyl...) Show SMILES Show InChI	GoogleScholar	UniChem		1.07E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily V member 1 (Human)	BDBM20461 (Zostrix | (E)-N-[(4-hydroxy-3-methoxyphenyl)methyl...) Show SMILES Show InChI	GoogleScholar	UniChem		1.14E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
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Transient receptor potential cation channel subfamily V member 1 (Rat)	BDBM20461 (Zostrix | (E)-N-[(4-hydroxy-3-methoxyphenyl)methyl...) Show SMILES Show InChI	GoogleScholar	UniChem		1.70E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily V member 1 (Rat)	BDBM20461 (Zostrix | (E)-N-[(4-hydroxy-3-methoxyphenyl)methyl...) Show SMILES Show InChI	GoogleScholar	UniChem		1.80E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Transient receptor potential cation channel subfamily V member 1 (Rat)	BDBM20461 (Zostrix | (E)-N-[(4-hydroxy-3-methoxyphenyl)methyl...) Show SMILES Show InChI	GoogleScholar	UniChem		1.81E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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