BDBM211264 US9247759, 10-12
SMILES Cc1noc(C)c1Cn1cc(cn1)N1C(=O)CN(Cc2ccc(O)cc2)C1=O
InChI Key InChIKey=RMCGUMMUZSKYJB-UHFFFAOYSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 211264
Affinity DataIC50: 40nMAssay Description:Antagonist activity at recombinant human TAS2R8 stably expressed in cells co-expressing Galpha16gust44 assessed as inhibition of andrographolide-indu...More data for this Ligand-Target Pair
Affinity DataIC50: 60nMAssay Description:In another embodiment, Fluorescence Polarization ("FP") based assays may be used to detect and monitor ligand binding. Fluorescence polarization is a...More data for this Ligand-Target Pair