BDBM21279 1-(2,4-dichlorophenyl)-5-(4-iodophenyl)-4-methyl-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide::AM 251::AM-251::AM251::CHEMBL285932::N-(piperidin-1-yl)-1-(2,4-dichlorophenyl)-5-(4-iodophenyl)-4-methyl-1H-pyrazole-3-carboxamide

SMILES: Cc1c(nn(c1-c1ccc(I)cc1)-c1ccc(Cl)cc1Cl)C(=O)NN1CCCCC1

InChI Key: InChIKey=BUZAJRPLUGXRAB-UHFFFAOYSA-N

Data: 20 KI  2 IC50  3 EC50

Find this compound or compounds like it in BindingDB or PDB:

Substructure Similarity at least:  must be >=0.5 Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 25 hits for monomerid = 21279   

Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50 nM	koff s-1	kon M-1s-1	pH	Temp °C
Cannabinoid receptor 1 (Human)	BDBM21279 (N-(piperidin-1-yl)-1-(2,4-dichlorophenyl)-5-(4-iod...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	0.320	n/a	n/a	n/a	n/a	n/a	n/a
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Cannabinoid receptor 1 (Human)	BDBM21279 (N-(piperidin-1-yl)-1-(2,4-dichlorophenyl)-5-(4-iod...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	3.5	n/a	n/a	n/a	n/a	n/a	n/a
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Cannabinoid receptor 1 (Human)	BDBM21279 (N-(piperidin-1-yl)-1-(2,4-dichlorophenyl)-5-(4-iod...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	n/a	68	n/a	n/a	n/a	n/a
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Cannabinoid receptor 1 (Human)	BDBM21279 (N-(piperidin-1-yl)-1-(2,4-dichlorophenyl)-5-(4-iod...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	n/a	58	n/a	n/a	n/a	n/a
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Cannabinoid receptor 1 (Human)	BDBM21279 (N-(piperidin-1-yl)-1-(2,4-dichlorophenyl)-5-(4-iod...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	n/a	70	n/a	n/a	n/a	n/a
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Cannabinoid receptor 1 (Rat)	BDBM21279 (N-(piperidin-1-yl)-1-(2,4-dichlorophenyl)-5-(4-iod...) Show SMILES Show InChI	GoogleScholar	UniChem		0.600	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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Cannabinoid receptor 1 (Human)	BDBM21279 (N-(piperidin-1-yl)-1-(2,4-dichlorophenyl)-5-(4-iod...) Show SMILES Show InChI	GoogleScholar	UniChem		2.30	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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					More data for this Ligand-Target Pair
Cannabinoid receptor 1 (Human)	BDBM21279 (N-(piperidin-1-yl)-1-(2,4-dichlorophenyl)-5-(4-iod...) Show SMILES Show InChI	GoogleScholar	UniChem		2.30	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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					More data for this Ligand-Target Pair
Cannabinoid receptor 1 (Human)	BDBM21279 (N-(piperidin-1-yl)-1-(2,4-dichlorophenyl)-5-(4-iod...) Show SMILES Show InChI	GoogleScholar	UniChem		2.30	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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					More data for this Ligand-Target Pair
Cannabinoid receptor 1 (Human)	BDBM21279 (N-(piperidin-1-yl)-1-(2,4-dichlorophenyl)-5-(4-iod...) Show SMILES Show InChI	GoogleScholar	UniChem		2.30	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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Cannabinoid receptor 1 (Human)	BDBM21279 (N-(piperidin-1-yl)-1-(2,4-dichlorophenyl)-5-(4-iod...) Show SMILES Show InChI	GoogleScholar	UniChem		3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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Cannabinoid receptor 1 (Rat)	BDBM21279 (N-(piperidin-1-yl)-1-(2,4-dichlorophenyl)-5-(4-iod...) Show SMILES Show InChI	GoogleScholar	UniChem		6	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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					More data for this Ligand-Target Pair
Cannabinoid receptor 1 (Human)	BDBM21279 (N-(piperidin-1-yl)-1-(2,4-dichlorophenyl)-5-(4-iod...) Show SMILES Show InChI	GoogleScholar	UniChem		7.49	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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					More data for this Ligand-Target Pair
Cannabinoid receptor 1 (Rat)	BDBM21279 (N-(piperidin-1-yl)-1-(2,4-dichlorophenyl)-5-(4-iod...) Show SMILES Show InChI	GoogleScholar	UniChem		7.49	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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					More data for this Ligand-Target Pair
Cannabinoid receptor 1 (Rat)	BDBM21279 (N-(piperidin-1-yl)-1-(2,4-dichlorophenyl)-5-(4-iod...) Show SMILES Show InChI	GoogleScholar	UniChem		7.5	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Cannabinoid receptor 1 (Human)	BDBM21279 (N-(piperidin-1-yl)-1-(2,4-dichlorophenyl)-5-(4-iod...) Show SMILES Show InChI	GoogleScholar	UniChem		7.5	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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					More data for this Ligand-Target Pair
Cannabinoid receptor 1 (Human)	BDBM21279 (N-(piperidin-1-yl)-1-(2,4-dichlorophenyl)-5-(4-iod...) Show SMILES Show InChI	GoogleScholar	UniChem		7.5	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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Cannabinoid receptor 1/2 (Rat)	BDBM21279 (N-(piperidin-1-yl)-1-(2,4-dichlorophenyl)-5-(4-iod...) Show SMILES Show InChI	GoogleScholar	UniChem		69	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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					More data for this Ligand-Target Pair
Cannabinoid receptor 2 (Human)	BDBM21279 (N-(piperidin-1-yl)-1-(2,4-dichlorophenyl)-5-(4-iod...) Show SMILES Show InChI	GoogleScholar	UniChem		110	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Cannabinoid receptor 2 (Human)	BDBM21279 (N-(piperidin-1-yl)-1-(2,4-dichlorophenyl)-5-(4-iod...) Show SMILES Show InChI	GoogleScholar	UniChem		112	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Cannabinoid receptor 2 (Human)	BDBM21279 (N-(piperidin-1-yl)-1-(2,4-dichlorophenyl)-5-(4-iod...) Show SMILES Show InChI	GoogleScholar	UniChem		112	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Cannabinoid receptor 2 (Human)	BDBM21279 (N-(piperidin-1-yl)-1-(2,4-dichlorophenyl)-5-(4-iod...) Show SMILES Show InChI	GoogleScholar	UniChem		112	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Cannabinoid receptor 2 (Human)	BDBM21279 (N-(piperidin-1-yl)-1-(2,4-dichlorophenyl)-5-(4-iod...) Show SMILES Show InChI	GoogleScholar	UniChem		2.29E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Cannabinoid receptor 1 (Rat)	BDBM21279 (N-(piperidin-1-yl)-1-(2,4-dichlorophenyl)-5-(4-iod...) Show SMILES Show InChI	GoogleScholar	UniChem		2.29E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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					More data for this Ligand-Target Pair
Cannabinoid receptor 2 (Mouse)	BDBM21279 (N-(piperidin-1-yl)-1-(2,4-dichlorophenyl)-5-(4-iod...) Show SMILES Show InChI	GoogleScholar	UniChem		2.29E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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					More data for this Ligand-Target Pair