BindingDB BDBM21280 5-(4-chloro-3-methylphenyl)-1-[(4-methylphenyl)methyl]-N-[(1S)-1,3,3-trimethylbicyclo[2.2.1]heptan-2-yl]-1H-pyrazole-3-carboxamide::N-(1,3,3-trimethylbicyclo(2.2.1)heptan-2-yl)-5-(4-chloro-3-methylphenyl)-1-(4-methylbenzyl)pyrazole-3-carboxamide::SR 144528::SR-144528::SR144528

BDBM21280 5-(4-chloro-3-methylphenyl)-1-[(4-methylphenyl)methyl]-N-[(1S)-1,3,3-trimethylbicyclo[2.2.1]heptan-2-yl]-1H-pyrazole-3-carboxamide::N-(1,3,3-trimethylbicyclo(2.2.1)heptan-2-yl)-5-(4-chloro-3-methylphenyl)-1-(4-methylbenzyl)pyrazole-3-carboxamide::SR 144528::SR-144528::SR144528

SMILES Cc1ccc(Cn2nc(cc2-c2ccc(Cl)c(C)c2)C(=O)NC2[C@@]3(C)CCC(C3)C2(C)C)cc1

InChI Key InChIKey=SUGVYNSRNKFXQM-ACSDJOOWSA-N

Data 83 KI

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 83 hits for monomerid = 21280

Cannabinoid receptor 2(MOUSE)
Japan Tobacco

Curated by PDSP K_i Database

PNG

BDBM21280(5-(4-chloro-3-methylphenyl)-1-[(4-methylphenyl)met...)

Ki: 0.0400nMMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

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Cannabinoid receptor 2(MOUSE)
Japan Tobacco

Curated by PDSP K_i Database

PNG

BDBM21280(5-(4-chloro-3-methylphenyl)-1-[(4-methylphenyl)met...)

Ki: 0.0500nMMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

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Cannabinoid receptor 2(Rattus norvegicus (Rat))
Japan Tobacco

Curated by PDSP K_i Database

PNG

BDBM21280(5-(4-chloro-3-methylphenyl)-1-[(4-methylphenyl)met...)

Ki: 0.240nMMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

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Cannabinoid receptor 2(Rattus norvegicus (Rat))
Japan Tobacco

Curated by PDSP K_i Database

PNG

BDBM21280(5-(4-chloro-3-methylphenyl)-1-[(4-methylphenyl)met...)

Ki: 0.300nMMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

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Cannabinoid receptor 2(Rattus norvegicus (Rat))
Japan Tobacco

Curated by PDSP K_i Database

PNG

BDBM21280(5-(4-chloro-3-methylphenyl)-1-[(4-methylphenyl)met...)

Ki: 0.300nMMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

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Cannabinoid receptor 2(Homo sapiens (Human))
Virginia Commonwealth University

Curated by PDSP K_i Database

PNG

BDBM21280(5-(4-chloro-3-methylphenyl)-1-[(4-methylphenyl)met...)

Ki: 0.320nMMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt UniProtKB/TrEMBL
DrugBank antibodypedia GoogleScholar

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Cannabinoid receptor 2(Homo sapiens (Human))
Virginia Commonwealth University

Curated by PDSP K_i Database

PNG

BDBM21280(5-(4-chloro-3-methylphenyl)-1-[(4-methylphenyl)met...)

Ki: 0.600nMMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt UniProtKB/TrEMBL
DrugBank antibodypedia GoogleScholar

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Cannabinoid receptor 2(Homo sapiens (Human))
Virginia Commonwealth University

Curated by PDSP K_i Database

PNG

BDBM21280(5-(4-chloro-3-methylphenyl)-1-[(4-methylphenyl)met...)

Ki: 1.99nMMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt UniProtKB/TrEMBL
DrugBank antibodypedia GoogleScholar

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Cannabinoid receptor 2(Homo sapiens (Human))
Virginia Commonwealth University

Curated by PDSP K_i Database

PNG

BDBM21280(5-(4-chloro-3-methylphenyl)-1-[(4-methylphenyl)met...)

Ki: 5.40nMAssay Description:IC50 values for test compounds were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibition c...More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt UniProtKB/TrEMBL
DrugBank antibodypedia GoogleScholar

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Details Article PubMed

Cannabinoid receptor 1(Mus musculus (Mouse))
Japan Tobacco

Curated by PDSP K_i Database

PNG

BDBM21280(5-(4-chloro-3-methylphenyl)-1-[(4-methylphenyl)met...)

Ki: 20.1nMMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
GoogleScholar

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Cannabinoid receptor 1(Rattus norvegicus (rat))
Japan Tobacco

Curated by PDSP K_i Database

PNG

BDBM21280(5-(4-chloro-3-methylphenyl)-1-[(4-methylphenyl)met...)

Ki: 27.6nMMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

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Cannabinoid receptor 1(Homo sapiens (Human))
Japan Tobacco

Curated by PDSP K_i Database

PNG

BDBM21280(5-(4-chloro-3-methylphenyl)-1-[(4-methylphenyl)met...)

Ki: 50.3nMMore data for this Ligand-Target Pair

PDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt UniProtKB/TrEMBL
DrugBank antibodypedia GoogleScholar

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Cannabinoid receptor 1(Rattus norvegicus (rat))
Japan Tobacco

Curated by PDSP K_i Database

PNG

BDBM21280(5-(4-chloro-3-methylphenyl)-1-[(4-methylphenyl)met...)

Ki: 305nMMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar

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Cannabinoid receptor 1(Homo sapiens (Human))
Japan Tobacco

Curated by PDSP K_i Database

PNG

BDBM21280(5-(4-chloro-3-methylphenyl)-1-[(4-methylphenyl)met...)

Ki: 437nMMore data for this Ligand-Target Pair

PDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt UniProtKB/TrEMBL
DrugBank antibodypedia GoogleScholar

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Cannabinoid receptor 1(Homo sapiens (Human))
Japan Tobacco

Curated by PDSP K_i Database

PNG

BDBM21280(5-(4-chloro-3-methylphenyl)-1-[(4-methylphenyl)met...)

Ki: >2.82E+3nMAssay Description:IC50 values for test compounds were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibition c...More data for this Ligand-Target Pair

PDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt UniProtKB/TrEMBL
DrugBank antibodypedia GoogleScholar

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Details Article PubMed

Pro-thyrotropin-releasing hormone(Homo sapiens (Human))
Sanofi Recherche

Curated by PDSP K_i Database

PNG

BDBM21280(5-(4-chloro-3-methylphenyl)-1-[(4-methylphenyl)met...)

Ki: >1.00E+4nMMore data for this Ligand-Target Pair

Reactome pathway KEGG
UniProtKB/SwissProt
antibodypedia GoogleScholar

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Vasopressin V1b receptor(Homo sapiens (Human))
Sanofi Recherche

Curated by PDSP K_i Database

PNG

BDBM21280(5-(4-chloro-3-methylphenyl)-1-[(4-methylphenyl)met...)

Ki: >1.00E+4nMMore data for this Ligand-Target Pair

Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

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Vasopressin V2 receptor(Homo sapiens (Human))
Sanofi Recherche

Curated by PDSP K_i Database

PNG

BDBM21280(5-(4-chloro-3-methylphenyl)-1-[(4-methylphenyl)met...)

Ki: >1.00E+4nMMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

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VIP peptides(Homo sapiens (Human))
Sanofi Recherche

Curated by PDSP K_i Database

PNG

BDBM21280(5-(4-chloro-3-methylphenyl)-1-[(4-methylphenyl)met...)

Ki: >1.00E+4nMMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

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5-hydroxytryptamine receptor 1B(Homo sapiens (Human))
Sanofi Recherche

Curated by PDSP K_i Database

PNG

BDBM21280(5-(4-chloro-3-methylphenyl)-1-[(4-methylphenyl)met...)

Ki: >1.00E+4nMMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

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5-hydroxytryptamine receptor 1D(Homo sapiens (Human))
Sanofi Recherche

Curated by PDSP K_i Database

PNG

BDBM21280(5-(4-chloro-3-methylphenyl)-1-[(4-methylphenyl)met...)

Ki: >1.00E+4nMMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

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5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Sanofi Recherche

Curated by PDSP K_i Database

PNG

BDBM21280(5-(4-chloro-3-methylphenyl)-1-[(4-methylphenyl)met...)

Ki: >1.00E+4nMMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

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5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Sanofi Recherche

Curated by PDSP K_i Database

PNG

BDBM21280(5-(4-chloro-3-methylphenyl)-1-[(4-methylphenyl)met...)

Ki: >1.00E+4nMMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

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5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Sanofi Recherche

Curated by PDSP K_i Database

PNG

BDBM21280(5-(4-chloro-3-methylphenyl)-1-[(4-methylphenyl)met...)

Ki: >1.00E+4nMMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

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5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Sanofi Recherche

Curated by PDSP K_i Database

PNG

BDBM21280(5-(4-chloro-3-methylphenyl)-1-[(4-methylphenyl)met...)

Ki: >1.00E+4nMMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

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Adenosine receptor A1(Homo sapiens (Human))
Sanofi Recherche

Curated by PDSP K_i Database

PNG

BDBM21280(5-(4-chloro-3-methylphenyl)-1-[(4-methylphenyl)met...)

Ki: >1.00E+4nMMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

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Adenosine receptor A2a(Homo sapiens (Human))
Sanofi Recherche

Curated by PDSP K_i Database

PNG

BDBM21280(5-(4-chloro-3-methylphenyl)-1-[(4-methylphenyl)met...)

Ki: >1.00E+4nMMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

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Alpha-1A adrenergic receptor(Homo sapiens (Human))
Sanofi Recherche

Curated by PDSP K_i Database

PNG

BDBM21280(5-(4-chloro-3-methylphenyl)-1-[(4-methylphenyl)met...)

Ki: >1.00E+4nMMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

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Alpha-2A adrenergic receptor(Homo sapiens (Human))
Sanofi Recherche

Curated by PDSP K_i Database

PNG

BDBM21280(5-(4-chloro-3-methylphenyl)-1-[(4-methylphenyl)met...)

Ki: >1.00E+4nMMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

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Beta-1 adrenergic receptor(Homo sapiens (Human))
Sanofi Recherche

Curated by PDSP K_i Database

PNG

BDBM21280(5-(4-chloro-3-methylphenyl)-1-[(4-methylphenyl)met...)

Ki: >1.00E+4nMMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

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Beta-2 adrenergic receptor(Homo sapiens (Human))
Sanofi Recherche

Curated by PDSP K_i Database

PNG

BDBM21280(5-(4-chloro-3-methylphenyl)-1-[(4-methylphenyl)met...)

Ki: >1.00E+4nMMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

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Type-1 angiotensin II receptor(Homo sapiens (Human))
Sanofi Recherche

Curated by PDSP K_i Database

PNG

BDBM21280(5-(4-chloro-3-methylphenyl)-1-[(4-methylphenyl)met...)

Ki: >1.00E+4nMMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

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B1 bradykinin receptor(Homo sapiens (Human))
Sanofi Recherche

Curated by PDSP K_i Database

PNG

BDBM21280(5-(4-chloro-3-methylphenyl)-1-[(4-methylphenyl)met...)

Ki: >1.00E+4nMMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
antibodypedia GoogleScholar

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B2 bradykinin receptor(Homo sapiens (Human))
Sanofi Recherche

Curated by PDSP K_i Database

PNG

BDBM21280(5-(4-chloro-3-methylphenyl)-1-[(4-methylphenyl)met...)

Ki: >1.00E+4nMMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

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Gamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
Sanofi Recherche

Curated by PDSP K_i Database

PNG

BDBM21280(5-(4-chloro-3-methylphenyl)-1-[(4-methylphenyl)met...)

Ki: >1.00E+4nMMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

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Peripheral-type benzodiazepine receptor-associated protein 1(Homo sapiens (Human))
Sanofi Recherche

Curated by PDSP K_i Database

PNG

BDBM21280(5-(4-chloro-3-methylphenyl)-1-[(4-methylphenyl)met...)

Ki: >1.00E+4nMMore data for this Ligand-Target Pair

Reactome pathway
UniProtKB/SwissProt
GoogleScholar

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Protein phosphatase 3 catalytic subunit alpha(Homo sapiens (Human))
Sanofi Recherche

Curated by PDSP K_i Database

PNG

BDBM21280(5-(4-chloro-3-methylphenyl)-1-[(4-methylphenyl)met...)

Ki: >1.00E+4nMMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

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Voltage-dependent L-type calcium channel subunit alpha-1C(Homo sapiens (Human))
Sanofi Recherche

Curated by PDSP K_i Database

PNG

BDBM21280(5-(4-chloro-3-methylphenyl)-1-[(4-methylphenyl)met...)

Ki: >1.00E+4nMMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

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Voltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Sanofi Recherche

Curated by PDSP K_i Database

PNG

BDBM21280(5-(4-chloro-3-methylphenyl)-1-[(4-methylphenyl)met...)

Ki: >1.00E+4nMMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

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Calpain-2 catalytic subunit(Homo sapiens (Human))
Sanofi Recherche

Curated by PDSP K_i Database

PNG

BDBM21280(5-(4-chloro-3-methylphenyl)-1-[(4-methylphenyl)met...)

Ki: >1.00E+4nMMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

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Gastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Sanofi Recherche

Curated by PDSP K_i Database

PNG

BDBM21280(5-(4-chloro-3-methylphenyl)-1-[(4-methylphenyl)met...)

Ki: >1.00E+4nMMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

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Gastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Sanofi Recherche

Curated by PDSP K_i Database

PNG

BDBM21280(5-(4-chloro-3-methylphenyl)-1-[(4-methylphenyl)met...)

Ki: >1.00E+4nMMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

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Muscarinic acetylcholine receptor M1(Homo sapiens (Human))
Sanofi Recherche

Curated by PDSP K_i Database

PNG

BDBM21280(5-(4-chloro-3-methylphenyl)-1-[(4-methylphenyl)met...)

Ki: >1.00E+4nMMore data for this Ligand-Target Pair

Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

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Muscarinic acetylcholine receptor M2(Homo sapiens (Human))
Sanofi Recherche

Curated by PDSP K_i Database

PNG

BDBM21280(5-(4-chloro-3-methylphenyl)-1-[(4-methylphenyl)met...)

Ki: >1.00E+4nMMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

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Muscarinic acetylcholine receptor M4(Homo sapiens (Human))
Sanofi Recherche

Curated by PDSP K_i Database

PNG

BDBM21280(5-(4-chloro-3-methylphenyl)-1-[(4-methylphenyl)met...)

Ki: >1.00E+4nMMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

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D(1A) dopamine receptor(Homo sapiens (Human))
Sanofi Recherche

Curated by PDSP K_i Database

PNG

BDBM21280(5-(4-chloro-3-methylphenyl)-1-[(4-methylphenyl)met...)

Ki: >1.00E+4nMMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

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D(2) dopamine receptor(Homo sapiens (Human))
Sanofi Recherche

Curated by PDSP K_i Database

PNG

BDBM21280(5-(4-chloro-3-methylphenyl)-1-[(4-methylphenyl)met...)

Ki: >1.00E+4nMMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

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D(3) dopamine receptor(Homo sapiens (Human))
Sanofi Recherche

Curated by PDSP K_i Database

PNG

BDBM21280(5-(4-chloro-3-methylphenyl)-1-[(4-methylphenyl)met...)

Ki: >1.00E+4nMMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

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D(4) dopamine receptor(Homo sapiens (Human))
Sanofi Recherche

Curated by PDSP K_i Database

PNG

BDBM21280(5-(4-chloro-3-methylphenyl)-1-[(4-methylphenyl)met...)

Ki: >1.00E+4nMMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

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Pro-epidermal growth factor(Homo sapiens (Human))
Sanofi Recherche

Curated by PDSP K_i Database

PNG

BDBM21280(5-(4-chloro-3-methylphenyl)-1-[(4-methylphenyl)met...)

Ki: >1.00E+4nMMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

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Displayed 1 to 50 (of 83 total ) | Next | Last >>

Filter my 83 hits

Targets 67▿
- Cannabinoid receptor 2 9
- Cannabinoid receptor 1 6
- Gastrin/cholecystokinin type B receptor 2
- Gamma-aminobutyric acid receptor subunit alpha-1 2
- Glutamate receptor ionotropic, NMDA 1 2
- Gamma-aminobutyric acid type B receptor subunit 1 1
- P2X purinoceptor 1 1
- Endothelin-1 receptor 1
- Galanin peptides 1
- Pro-epidermal growth factor 1
- Potassium voltage-gated channel subfamily A member 1 1
- Muscarinic acetylcholine receptor M4 1
- Muscarinic acetylcholine receptor M2 1
- Muscarinic acetylcholine receptor M1 1
- Beta-2 adrenergic receptor 1
- D(4) dopamine receptor 1
- Vasopressin V1b receptor 1
- Beta-1 adrenergic receptor 1
- D(2) dopamine receptor 1
- 5-hydroxytryptamine receptor 3A 1
- Neurotensin/neuromedin N 1
- Alpha-1A adrenergic receptor 1
- Voltage-dependent N-type calcium channel subunit alpha-1B 1
- Neuronal acetylcholine receptor subunit alpha-3 1
- Protein phosphatase 3 catalytic subunit alpha 1
- B2 bradykinin receptor 1
- Glutamate receptor 3 1
- ATP-sensitive inward rectifier potassium channel 1 1
- 5-hydroxytryptamine receptor 2C 1
- 5-hydroxytryptamine receptor 2A 1
- D(1A) dopamine receptor 1
- 5-hydroxytryptamine receptor 4 1
- Sodium channel protein type 1 subunit alpha 1
- Sodium channel protein type 2 subunit alpha 1
- Calpain-2 catalytic subunit 1
- B1 bradykinin receptor 1
- Platelet-activating factor receptor 1
- Substance-K receptor 1
- Adenosine receptor A1 1
- D(3) dopamine receptor 1
- Vasopressin V2 receptor 1
- Histamine H1 receptor 1
- 5-hydroxytryptamine receptor 1B 1
- Somatostatin 1
- Voltage-dependent L-type calcium channel subunit alpha-1C 1
- 5-hydroxytryptamine receptor 1D 1
- Thromboxane A2 receptor 1
- Substance-P receptor 1
- Histamine H3 receptor 1
- Protein kinase C beta type 1
- Leukotriene B4 receptor 2 1
- Neuropeptide Y receptor type 1 1
- Protein kinase C alpha type 1
- Neuropeptide Y receptor type 2 1
- Neuromedin-K receptor 1
- Pro-thyrotropin-releasing hormone 1
- Peripheral-type benzodiazepine receptor-associated protein 1 1
- Type-1 angiotensin II receptor 1
- Glutamate receptor ionotropic, kainate 1 1
- P2Y purinoceptor 1 1
- VIP peptides 1
- Calcium-activated potassium channel subunit beta-1 1
- AP-4 complex subunit sigma-1 1
- Endothelin receptor type B 1
- Alpha-2A adrenergic receptor 1
- Histamine H2 receptor 1
- Adenosine receptor A2a 1
Publications 4▿
- J Pharmacol Exp Ther 284: 644-50 (1998) 72
- J Pharmacol Exp Ther 296: 420-5 (2001) 6
- J Pharmacol Exp Ther 292: 886-94 (2000) 3
- J Med Chem 51: 1560-76 (2008) 2
Institutions 4▿
- Sanofi Recherche 72
- Japan Tobacco 6
- Virginia Commonwealth University 3
- Sapienza University Of Rome 2
Affinity: 0.040 to 1.0E+4 nM▿
- Ki 83
- Affinity ≤ nM
Xtal structures: 0
Docked structures: 0
Catalog Cmpds: 1