BDBM220447 US10633379, Compound X::US9296741, 36

SMILES: CCS(=O)(=O)Nc1ccc(c(c1)C2=CN(C(=O)c3c2cc[nH]3)C)Oc4ccc(cc4F)F

InChI Key: InChIKey=RDONXGFGWSSFMY-UHFFFAOYSA-N

Data: 10 KI  17 IC50  19 Kd  1 EC50

PDB links: 1 PDB ID matches this monomer.

Find this compound or compounds like it in BindingDB or PDB:

Substructure Similarity at least:  must be >=0.5 Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 49 hits for monomerid = 220447   

Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50 nM	koff s-1	kon M-1s-1	pH	Temp °C
Bromodomain-containing protein 4 (Human)	BDBM220447 (US9296741, 36 | US10633379, Compound X) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	20	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
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Protein polybromo-1 (Human)	BDBM220447 (US9296741, 36 | US10633379, Compound X) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	>1.00E+3	n/a	n/a	n/a	n/a	n/a
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Adenosine receptor A2b (Human)	BDBM220447 (US9296741, 36 | US10633379, Compound X) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	2.60E+3	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
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Histone acetyltransferase p300 (Human)	BDBM220447 (US9296741, 36 | US10633379, Compound X) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	87	n/a	n/a	n/a	n/a	n/a
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Peregrin (Human)	BDBM220447 (US9296741, 36 | US10633379, Compound X) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	>1.00E+3	n/a	n/a	n/a	n/a	n/a
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E3 ubiquitin-protein ligase TRIM33 (Human)	BDBM220447 (US9296741, 36 | US10633379, Compound X) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	>1.00E+3	n/a	n/a	n/a	n/a	n/a
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Bromodomain-containing protein 4 (Human)	BDBM220447 (US9296741, 36 | US10633379, Compound X) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	69	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Bromodomain-containing protein 4 (Human)	BDBM220447 (US9296741, 36 | US10633379, Compound X) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	74	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Bromodomain-containing protein 4 (Human)	BDBM220447 (US9296741, 36 | US10633379, Compound X) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	1	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Bromodomain-containing protein 4 (Human)	BDBM220447 (US9296741, 36 | US10633379, Compound X) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	20	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Bromodomain-containing protein 4 (Human)	BDBM220447 (US9296741, 36 | US10633379, Compound X) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	39	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Bromodomain-containing protein 4 (Human)	BDBM220447 (US9296741, 36 | US10633379, Compound X) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	47	n/a	n/a	n/a	n/a	n/a	n/a
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Transcription intermediary factor 1-alpha (Human)	BDBM220447 (US9296741, 36 | US10633379, Compound X) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	>1.00E+3	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Histone acetyltransferase p300 (Human)	BDBM220447 (US9296741, 36 | US10633379, Compound X) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	63	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Bromodomain-containing protein 4 (Human)	BDBM220447 (US9296741, 36 | US10633379, Compound X) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	2.70	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Bromodomain-containing protein 4 (Human)	BDBM220447 (US9296741, 36 | US10633379, Compound X) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	1	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Bromodomain-containing protein 4 (Human)	BDBM220447 (US9296741, 36 | US10633379, Compound X) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	2.5	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Bromodomain-containing protein 4 (Human)	BDBM220447 (US9296741, 36 | US10633379, Compound X) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	11	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Bromodomain-containing protein 4 (Human)	BDBM220447 (US9296741, 36 | US10633379, Compound X) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	3	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Bromodomain-containing protein 4 (Human)	BDBM220447 (US9296741, 36 | US10633379, Compound X) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	3	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Bromodomain-containing protein 4 (Human)	BDBM220447 (US9296741, 36 | US10633379, Compound X) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	0.700	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Bromodomain-containing protein 4 (Human)	BDBM220447 (US9296741, 36 | US10633379, Compound X) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	14	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Bromodomain-containing protein 4 (Human)	BDBM220447 (US9296741, 36 | US10633379, Compound X) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	3	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Transcription activator BRG1 (Human)	BDBM220447 (US9296741, 36 | US10633379, Compound X) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	>1.00E+3	n/a	n/a	n/a	n/a	n/a
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Bromodomain-containing protein 8 (Human)	BDBM220447 (US9296741, 36 | US10633379, Compound X) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	>1.00E+3	n/a	n/a	n/a	n/a	n/a
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Bromodomain adjacent to zinc finger domain protein 2A (Human)	BDBM220447 (US9296741, 36 | US10633379, Compound X) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	>1.00E+3	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
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Bromodomain adjacent to zinc finger domain protein 2B (Human)	BDBM220447 (US9296741, 36 | US10633379, Compound X) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	>1.00E+3	n/a	n/a	n/a	n/a	n/a
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Bromodomain and PHD finger-containing protein 3 (Human)	BDBM220447 (US9296741, 36 | US10633379, Compound X) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	>1.00E+3	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Protein polybromo-1 (Human)	BDBM220447 (US9296741, 36 | US10633379, Compound X) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	>1.00E+3	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
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Bromodomain and WD repeat-containing protein 1 (Human)	BDBM220447 (US9296741, 36 | US10633379, Compound X) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	>1.00E+3	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Bromodomain-containing protein 4 (Human)	BDBM220447 (US9296741, 36 | US10633379, Compound X) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	n/a	20	n/a	n/a	n/a	n/a
TBA									Citation and Details
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Transcription initiation factor TFIID subunit 1-like (Human)	BDBM220447 (US9296741, 36 | US10633379, Compound X) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	>1.00E+3	n/a	n/a	n/a	n/a	n/a
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Bromodomain-containing protein 7 (Human)	BDBM220447 (US9296741, 36 | US10633379, Compound X) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	>1.00E+3	n/a	n/a	n/a	n/a	n/a
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Histone acetyltransferase KAT2B (Human)	BDBM220447 (US9296741, 36 | US10633379, Compound X) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	>1.00E+3	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
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Histone acetyltransferase KAT2A (Human)	BDBM220447 (US9296741, 36 | US10633379, Compound X) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	>1.00E+3	n/a	n/a	n/a	n/a	n/a
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Chromatin remodeling regulator CECR2 (Human)	BDBM220447 (US9296741, 36 | US10633379, Compound X) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	>1.00E+3	n/a	n/a	n/a	n/a	n/a
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Translocator protein (Human)	BDBM220447 (US9296741, 36 | US10633379, Compound X) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	800	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Bromodomain-containing protein 4 (Human)	BDBM220447 (US9296741, 36 | US10633379, Compound X) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	<10	n/a	n/a	n/a	n/a	n/a
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Bromodomain-containing protein 9 (Human)	BDBM220447 (US9296741, 36 | US10633379, Compound X) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	>1.00E+3	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
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Bromodomain-containing protein 4 [352-457] (Human)	BDBM220447 (US9296741, 36 | US10633379, Compound X) Show SMILES Show InChI	GoogleScholar	UniChem		0.952	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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Bromodomain-containing protein 2 (Human)	BDBM220447 (US9296741, 36 | US10633379, Compound X) Show SMILES Show InChI	GoogleScholar	UniChem		1	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Bromodomain-containing protein 4 [352-457] (Human)	BDBM220447 (US9296741, 36 | US10633379, Compound X) Show SMILES Show InChI	GoogleScholar	UniChem		1.40	-12.1	n/a	n/a	n/a	n/a	n/a	6.0	25
TBA									Citation and Details
					More data for this Ligand-Target Pair
Bromodomain-containing protein 4 (Human)	BDBM220447 (US9296741, 36 | US10633379, Compound X) Show SMILES Show InChI	GoogleScholar	UniChem		1.5	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Bromodomain-containing protein 4 (Human)	BDBM220447 (US9296741, 36 | US10633379, Compound X) Show SMILES Show InChI	GoogleScholar	UniChem		1.5	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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Bromodomain-containing protein 4 [57-168] (Human)	BDBM220447 (US9296741, 36 | US10633379, Compound X) Show SMILES Show InChI	GoogleScholar	UniChem		2.09	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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Bromodomain testis-specific protein (Human)	BDBM220447 (US9296741, 36 | US10633379, Compound X) Show SMILES Show InChI	GoogleScholar	UniChem		2.20	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Bromodomain-containing protein 4 [57-168] (Human)	BDBM220447 (US9296741, 36 | US10633379, Compound X) Show SMILES Show InChI	GoogleScholar	UniChem		3.5	-11.5	n/a	n/a	n/a	n/a	n/a	6.0	25
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Bromodomain-containing protein 3 (Human)	BDBM220447 (US9296741, 36 | US10633379, Compound X) Show SMILES Show InChI	GoogleScholar	UniChem		12	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Bromodomain-containing protein 4 (Human)	BDBM220447 (US9296741, 36 | US10633379, Compound X) Show SMILES Show InChI	GoogleScholar	UniChem		15	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair