BDBM228250 N-((1s,4s)-4-(3-methyl-8-(6-(1-methyl-1H-pyrazol-4-yl)pyridin-3-yl)-2-oxo-2,3-dihydro-1H-imidazo[4,5-c]quinolin-1-yl)cyclohexyl)acetamide::US10047084, 33

SMILES CC(=O)N[C@H]1CC[C@H](CC1)n1c2c(cnc3ccc(cc23)-c2ccc(nc2)-c2cnn(C)c2)n(C)c1=O

InChI Key InChIKey=AQXKYGUPFRNYIE-SZPZYZBQSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
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Similarity at least:  must be >=0.5
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 228250   

TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Beijing Forelandpharma

US Patent
LigandPNGBDBM228250(N-((1s,4s)-4-(3-methyl-8-(6-(1-methyl-1H-pyrazol-4...)
Affinity DataIC50: <10nMAssay Description:The inhibition of the mTOR protein kinase activity by the compounds was determined by the enzymatic activity assay in vitro. The detection kit suppli...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent