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BDBM22877 2-((1-(1-(4-fluorobenzyl)-1H-benzo[d]imidazol-2-yl)piperidin-4-yl)(methyl)amino)pyrimidin-4(3H)-one::2-({1-[1-(4-Fluoro-benzyl)-1H-benzoimidazol-2-yl]-piperidin-4-yl}-methyl-amino)-3H-pyrimidin-4-one::2-({1-[3-(4-Fluoro-benzyl)-1H-benzoimidazol-2-yl]-piperidin-4-yl}-methyl-amino)-2,3-dihydro-1H-pyrimidin-4-one(Mizolastine)::2-[(1-{1-[(4-fluorophenyl)methyl]-1H-1,3-benzodiazol-2-yl}piperidin-4-yl)(methyl)amino]-3,4-dihydropyrimidin-4-one::CHEMBL94454::Mizolastine::Mizollen::Zolistan

SMILES: CN(C1CCN(CC1)c1nc2ccccc2n1Cc1ccc(F)cc1)c1nccc(=O)[nH]1

InChI Key: InChIKey=PVLJETXTTWAYEW-UHFFFAOYSA-N

Data: 5 KI  9 IC50

Find this compound or compounds like it in BindingDB or PDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 14 hits for monomerid = 22877   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kcal/mole
IC50
nM
Kd
nM
EC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Cytochrome P450 3A4


(Human)
BDBM22877
PNG
(Zolistan | 2-[(1-{1-[(4-fluorophenyl)methyl]-1H-1,...)
GoogleScholar
UniChem
n/an/a>5.00E+3n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Potassium voltage-gated channel subfamily H member 2


(Human)
BDBM22877
PNG
(Zolistan | 2-[(1-{1-[(4-fluorophenyl)methyl]-1H-1,...)
GoogleScholar
UniChem
n/an/a 441n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Potassium voltage-gated channel subfamily H member 2


(Human)
BDBM22877
PNG
(Zolistan | 2-[(1-{1-[(4-fluorophenyl)methyl]-1H-1,...)
GoogleScholar
UniChem
n/an/a 437n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Potassium voltage-gated channel subfamily H member 2


(Human)
BDBM22877
PNG
(Zolistan | 2-[(1-{1-[(4-fluorophenyl)methyl]-1H-1,...)
GoogleScholar
UniChem
n/an/a 350n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Potassium voltage-gated channel subfamily H member 2


(Human)
BDBM22877
PNG
(Zolistan | 2-[(1-{1-[(4-fluorophenyl)methyl]-1H-1,...)
GoogleScholar
UniChem
n/an/a 437n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Potassium voltage-gated channel subfamily H member 2


(Human)
BDBM22877
PNG
(Zolistan | 2-[(1-{1-[(4-fluorophenyl)methyl]-1H-1,...)
GoogleScholar
UniChem
n/an/a 437n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Potassium voltage-gated channel subfamily H member 2


(Human)
BDBM22877
PNG
(Zolistan | 2-[(1-{1-[(4-fluorophenyl)methyl]-1H-1,...)
GoogleScholar
UniChem
n/an/a 355n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Potassium voltage-gated channel subfamily H member 2


(Human)
BDBM22877
PNG
(Zolistan | 2-[(1-{1-[(4-fluorophenyl)methyl]-1H-1,...)
GoogleScholar
UniChem
n/an/a 437n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Potassium voltage-gated channel subfamily H member 2


(Human)
BDBM22877
PNG
(Zolistan | 2-[(1-{1-[(4-fluorophenyl)methyl]-1H-1,...)
GoogleScholar
UniChem
n/an/a 355n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Histamine H1 receptor


(Human)
BDBM22877
PNG
(Zolistan | 2-[(1-{1-[(4-fluorophenyl)methyl]-1H-1,...)
GoogleScholar
UniChem
2.70n/an/an/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Potassium voltage-gated channel subfamily H member 2


(Human)
BDBM22877
PNG
(Zolistan | 2-[(1-{1-[(4-fluorophenyl)methyl]-1H-1,...)
GoogleScholar
UniChem
7.26E+3n/an/an/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Histamine H4 receptor


(Human)
BDBM22877
PNG
(Zolistan | 2-[(1-{1-[(4-fluorophenyl)methyl]-1H-1,...)
GoogleScholar
UniChem
>1.00E+4>-7.09n/an/an/an/an/a7.437


TBA



Citation and Details
More data for this
Ligand-Target Pair
Muscarinic acetylcholine receptor M1


(Human)
BDBM22877
PNG
(Zolistan | 2-[(1-{1-[(4-fluorophenyl)methyl]-1H-1,...)
GoogleScholar
UniChem
>1.00E+4n/an/an/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Cytochrome P450 2D6


(Human)
BDBM22877
PNG
(Zolistan | 2-[(1-{1-[(4-fluorophenyl)methyl]-1H-1,...)
GoogleScholar
UniChem
>2.00E+4n/an/an/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair