BDBM238766 US9394297, 450

SMILES: C[C@H]1NC(=O)c2cc([nH]c12)-c1cccc2c1nc(NC(C)(C)C)n(C)c2=O

InChI Key: InChIKey=HLPARXMUJBJYFM-UHFFFAOYSA-N

Data: 12 IC50  3 Kd

Find this compound or compounds like it in BindingDB or PDB:

Substructure Similarity at least:  must be >=0.5 Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 15 hits for monomerid = 238766   

Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50 nM	koff s-1	kon M-1s-1	pH	Temp °C
Serine/threonine-protein kinase pim-1 (Human)	BDBM238766 (US9394297, 450) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	0.779	n/a	n/a	n/a	n/a	7.0	22
TBA									Citation and Details
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Serine/threonine-protein kinase pim-2 (Human)	BDBM238766 (US9394297, 450) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	0.826	n/a	n/a	n/a	n/a	7.0	22
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Serine/threonine-protein kinase pim-1 (Human)	BDBM238766 (US9394297, 450) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	0.340	n/a	n/a	n/a	n/a	n/a	n/a
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					More data for this Ligand-Target Pair
Serine/threonine-protein kinase pim-2 (Human)	BDBM238766 (US9394297, 450) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	0.380	n/a	n/a	n/a	n/a	n/a	n/a
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Cytochrome P450 3A4 (Human)	BDBM238766 (US9394297, 450) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	>5.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Serine/threonine-protein kinase pim-1 (Human)	BDBM238766 (US9394297, 450) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	0.300	n/a	n/a	n/a	n/a	n/a	n/a
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					More data for this Ligand-Target Pair
Serine/threonine-protein kinase pim-2 (Human)	BDBM238766 (US9394297, 450) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	0.200	n/a	n/a	n/a	n/a	n/a	n/a
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Serine/threonine-protein kinase pim-1/pim-2/pim-3 (Human)	BDBM238766 (US9394297, 450) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	31	n/a	n/a	n/a	n/a	n/a	n/a
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Cytochrome P450 2C19 (Human)	BDBM238766 (US9394297, 450) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	3.10E+4	n/a	n/a	n/a	n/a	n/a	n/a
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Cytochrome P450 2D6 (Human)	BDBM238766 (US9394297, 450) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	>5.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
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					More data for this Ligand-Target Pair
Serine/threonine-protein kinase pim-1 (Human)	BDBM238766 (US9394297, 450) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	1.30	n/a	n/a	n/a	n/a	n/a
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Cytochrome P450 1A2 (Human)	BDBM238766 (US9394297, 450) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	>5.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
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Serine/threonine-protein kinase pim-3 (Human)	BDBM238766 (US9394297, 450) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	1.20	n/a	n/a	n/a	n/a	n/a
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Potassium voltage-gated channel subfamily H member 2 (Human)	BDBM238766 (US9394297, 450) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	>3.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Serine/threonine-protein kinase pim-2 (Human)	BDBM238766 (US9394297, 450) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	1.70	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair