BDBM249277 US10017501, Compound 1020-18::US9458145, 1020-18

SMILES: Cc1noc(C)c1-c1cc(-c2c(C)ccc3ncccc23)c2[nH]c(nc2c1)C1CC1

InChI Key: InChIKey=KHQQNXFBTALTQF-UHFFFAOYSA-N

Data: 3 KI  7 IC50  40 Kd  1 EC50

Find this compound or compounds like it in BindingDB or PDB:

Substructure Similarity at least:  must be >=0.5 Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 51 hits for monomerid = 249277   

Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50 nM	koff s-1	kon M-1s-1	pH	Temp °C
Bromodomain-containing protein 3 (Human)	BDBM249277 (US9458145, 1020-18 | US10017501, Compound 1020-18) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	0.650	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
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Histone acetyltransferase KAT2A (Human)	BDBM249277 (US9458145, 1020-18 | US10017501, Compound 1020-18) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
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Protein polybromo-1 (Human)	BDBM249277 (US9458145, 1020-18 | US10017501, Compound 1020-18) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a
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Histone acetyltransferase KAT2B (Human)	BDBM249277 (US9458145, 1020-18 | US10017501, Compound 1020-18) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a
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Transcription activator BRG1 (Human)	BDBM249277 (US9458145, 1020-18 | US10017501, Compound 1020-18) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a
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Transcription initiation factor TFIID subunit 1 (Human)	BDBM249277 (US9458145, 1020-18 | US10017501, Compound 1020-18) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	8.00E+3	n/a	n/a	n/a	n/a	n/a
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Transcription intermediary factor 1-alpha (Human)	BDBM249277 (US9458145, 1020-18 | US10017501, Compound 1020-18) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	6.90E+3	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Bromodomain and WD repeat-containing protein 1 (Human)	BDBM249277 (US9458145, 1020-18 | US10017501, Compound 1020-18) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a
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Bromodomain-containing protein 2 (Human)	BDBM249277 (US9458145, 1020-18 | US10017501, Compound 1020-18) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	1.10	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Bromodomain-containing protein 4 (Human)	BDBM249277 (US9458145, 1020-18 | US10017501, Compound 1020-18) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	2.80	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Bromodomain and PHD finger-containing protein 3 (Human)	BDBM249277 (US9458145, 1020-18 | US10017501, Compound 1020-18) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a
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Probable global transcription activator SNF2L2 (Human)	BDBM249277 (US9458145, 1020-18 | US10017501, Compound 1020-18) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Bromodomain-containing protein 2 (Human)	BDBM249277 (US9458145, 1020-18 | US10017501, Compound 1020-18) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	2.5	n/a	n/a	n/a	n/a	n/a
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Chromatin remodeling regulator CECR2 (Human)	BDBM249277 (US9458145, 1020-18 | US10017501, Compound 1020-18) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	8.20E+3	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
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Bromodomain-containing protein 8 (Human)	BDBM249277 (US9458145, 1020-18 | US10017501, Compound 1020-18) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a
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Bromodomain testis-specific protein (Human)	BDBM249277 (US9458145, 1020-18 | US10017501, Compound 1020-18) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	4.90	n/a	n/a	n/a	n/a	n/a
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Nucleosome-remodeling factor subunit BPTF (Human)	BDBM249277 (US9458145, 1020-18 | US10017501, Compound 1020-18) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a
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Protein polybromo-1 (Human)	BDBM249277 (US9458145, 1020-18 | US10017501, Compound 1020-18) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
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Transcription intermediary factor 1-alpha (Human)	BDBM249277 (US9458145, 1020-18 | US10017501, Compound 1020-18) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	4.10E+3	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Bromodomain-containing protein 4 (Human)	BDBM249277 (US9458145, 1020-18 | US10017501, Compound 1020-18) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	78	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Bromodomain-containing protein 4 (Human)	BDBM249277 (US9458145, 1020-18 | US10017501, Compound 1020-18) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	83	n/a	n/a	n/a	n/a	n/a	n/a
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ATPase family AAA domain-containing protein 2B (Human)	BDBM249277 (US9458145, 1020-18 | US10017501, Compound 1020-18) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Bromodomain-containing protein 4 (Human)	BDBM249277 (US9458145, 1020-18 | US10017501, Compound 1020-18) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	1.30	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
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CREB-binding protein (Human)	BDBM249277 (US9458145, 1020-18 | US10017501, Compound 1020-18) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	170	n/a	n/a	n/a	n/a	n/a
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E3 ubiquitin-protein ligase TRIM33 (Human)	BDBM249277 (US9458145, 1020-18 | US10017501, Compound 1020-18) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
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ATPase family AAA domain-containing protein 2 (Human)	BDBM249277 (US9458145, 1020-18 | US10017501, Compound 1020-18) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a
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Bromodomain-containing protein 4 [368-440] (Human)	BDBM249277 (US9458145, 1020-18 | US10017501, Compound 1020-18) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	78.6	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
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Bromodomain-containing protein 4 [75-147] (Human)	BDBM249277 (US9458145, 1020-18 | US10017501, Compound 1020-18) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	87.1	n/a	n/a	n/a	n/a	7.5	25
TBA									Citation and Details
					More data for this Ligand-Target Pair
Bromodomain-containing protein 4 [368-440] (Human)	BDBM249277 (US9458145, 1020-18 | US10017501, Compound 1020-18) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	78.6	n/a	n/a	n/a	n/a	7.5	25
TBA									Citation and Details
					More data for this Ligand-Target Pair
Bromodomain-containing protein 4 [75-147] (Human)	BDBM249277 (US9458145, 1020-18 | US10017501, Compound 1020-18) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	14.4	n/a	n/a	n/a	n/a	7.5	25
TBA									Citation and Details
					More data for this Ligand-Target Pair
Bromodomain-containing protein 4 (Human)	BDBM249277 (US9458145, 1020-18 | US10017501, Compound 1020-18) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	n/a	55	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Bromodomain-containing protein 2 (Human)	BDBM249277 (US9458145, 1020-18 | US10017501, Compound 1020-18) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	0.590	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
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Bromodomain-containing protein 8 (Human)	BDBM249277 (US9458145, 1020-18 | US10017501, Compound 1020-18) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	5.90E+3	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
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Histone acetyltransferase p300 (Human)	BDBM249277 (US9458145, 1020-18 | US10017501, Compound 1020-18) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	220	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
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Transcription initiation factor TFIID subunit 1-like (Human)	BDBM249277 (US9458145, 1020-18 | US10017501, Compound 1020-18) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Bromodomain-containing protein 4 [75-147] (Human)	BDBM249277 (US9458145, 1020-18 | US10017501, Compound 1020-18) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	87.1	n/a	n/a	n/a	n/a	n/a	n/a
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Bromodomain adjacent to zinc finger domain protein 2A (Human)	BDBM249277 (US9458145, 1020-18 | US10017501, Compound 1020-18) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
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Bromodomain adjacent to zinc finger domain protein 2B (Human)	BDBM249277 (US9458145, 1020-18 | US10017501, Compound 1020-18) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a
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					More data for this Ligand-Target Pair
Bromodomain-containing protein 1 (Human)	BDBM249277 (US9458145, 1020-18 | US10017501, Compound 1020-18) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a
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Bromodomain-containing protein 3 (Human)	BDBM249277 (US9458145, 1020-18 | US10017501, Compound 1020-18) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	1.70	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Bromodomain-containing protein 3 (Human)	BDBM249277 (US9458145, 1020-18 | US10017501, Compound 1020-18) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	0.660	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Bromodomain-containing protein 4 (Human)	BDBM249277 (US9458145, 1020-18 | US10017501, Compound 1020-18) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	2.90	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Bromodomain-containing protein 4 (Human)	BDBM249277 (US9458145, 1020-18 | US10017501, Compound 1020-18) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	3.20	n/a	n/a	n/a	n/a	n/a
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Bromodomain-containing protein 7 (Human)	BDBM249277 (US9458145, 1020-18 | US10017501, Compound 1020-18) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a
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Bromodomain-containing protein 9 (Human)	BDBM249277 (US9458145, 1020-18 | US10017501, Compound 1020-18) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a
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Bromodomain testis-specific protein (Human)	BDBM249277 (US9458145, 1020-18 | US10017501, Compound 1020-18) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	19	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Bromodomain testis-specific protein (Human)	BDBM249277 (US9458145, 1020-18 | US10017501, Compound 1020-18) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	5	n/a	n/a	n/a	n/a	n/a
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Peregrin (Human)	BDBM249277 (US9458145, 1020-18 | US10017501, Compound 1020-18) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	4.10E+3	n/a	n/a	n/a	n/a	n/a
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Bromodomain-containing protein 4 (Human)	BDBM249277 (US9458145, 1020-18 | US10017501, Compound 1020-18) Show SMILES Show InChI	GoogleScholar	UniChem		3.80	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Bromodomain-containing protein 4 (Human)	BDBM249277 (US9458145, 1020-18 | US10017501, Compound 1020-18) Show SMILES Show InChI	GoogleScholar	UniChem		7.5	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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					More data for this Ligand-Target Pair