BDBM25521 2-amino-pyrazolopyridine, 37::N-{2-[3-chloro-5-(3-methyl-6-{[(1S)-1-phenylethyl]amino}-1H-pyrazolo[4,3-c]pyridin-1-yl)phenyl]phenyl}acetamide
SMILES C[C@H](Nc1cc2n(nc(C)c2cn1)-c1cc(Cl)cc(c1)-c1ccccc1NC(C)=O)c1ccccc1
InChI Key InChIKey=QUYZXRAAIRZUEE-SFHVURJKSA-N
Data 5 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 5 hits for monomerid = 25521
Affinity DataIC50: 207nMpH: 7.2 T: 2°CAssay Description:An IMAP fluorescence polarization-based assay format (Molecular Devices) was used to determine the ability of compounds to inhibit the phosphorylatio...More data for this Ligand-Target Pair
Affinity DataIC50: 2.17E+3nMpH: 7.2 T: 2°CAssay Description:An IMAP fluorescence polarization-based assay format (Molecular Devices) was used to determine the ability of compounds to inhibit the phosphorylatio...More data for this Ligand-Target Pair
Affinity DataIC50: 6.28E+3nMAssay Description:The activity was measured by off-chip mobility shift assay. The enzyme was incubated with fluorecence-labeled peptide substrate and Mg(or Mn)/ATP. Th...More data for this Ligand-Target Pair
Affinity DataIC50: 6.80E+3nMAssay Description:The activity was determined by IMAP assay. The enzyme was incubated with fluorescein labeled peptide and phosphorylation was detected by IMAP technol...More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMpH: 7.2 T: 2°CAssay Description:An IMAP fluorescence polarization-based assay format (Molecular Devices) was used to determine the ability of compounds to inhibit the phosphorylatio...More data for this Ligand-Target Pair