BDBM255370 US9481682, 121

SMILES: Nc1nccn2c(nc(-c3ccc(cc3OC3CC3)C(=O)Nc3cc(ccn3)C(F)(F)F)c12)[C@@H]1CC[C@H]2CCC(=O)N2C1

InChI Key: InChIKey=WMMNTQFZCHUZSM-UHFFFAOYSA-N

Data: 20 IC50

Find this compound or compounds like it in BindingDB or PDB:

Substructure Similarity at least:  must be >=0.5 Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 20 hits for monomerid = 255370   

Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50 nM	koff s-1	kon M-1s-1	pH	Temp °C
Tyrosine-protein kinase Fyn (Human)	BDBM255370 (US9481682, 121) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	7.40E+3	n/a	n/a	n/a	n/a	n/a	n/a
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Tyrosine-protein kinase BTK (Human)	BDBM255370 (US9481682, 121) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	1.40	n/a	n/a	n/a	n/a	n/a	n/a
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Tyrosine-protein kinase Yes (Human)	BDBM255370 (US9481682, 121) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	430	n/a	n/a	n/a	n/a	n/a	n/a
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Tyrosine-protein kinase TXK (Human)	BDBM255370 (US9481682, 121) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	312	n/a	n/a	n/a	n/a	n/a	n/a
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Tyrosine-protein kinase Tec (Human)	BDBM255370 (US9481682, 121) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	277	n/a	n/a	n/a	n/a	n/a	n/a
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Tyrosine-protein kinase Srms (Human)	BDBM255370 (US9481682, 121) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	61	n/a	n/a	n/a	n/a	n/a	n/a
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Proto-oncogene tyrosine-protein kinase Src (Human)	BDBM255370 (US9481682, 121) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	946	n/a	n/a	n/a	n/a	n/a	n/a
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Protein-tyrosine kinase 6 (Human)	BDBM255370 (US9481682, 121) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	320	n/a	n/a	n/a	n/a	n/a	n/a
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Tyrosine-protein kinase Lyn (Human)	BDBM255370 (US9481682, 121) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	865	n/a	n/a	n/a	n/a	n/a	n/a
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Tyrosine-protein kinase Lck (Human)	BDBM255370 (US9481682, 121) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	182	n/a	n/a	n/a	n/a	n/a	n/a
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Tyrosine-protein kinase BTK (Human)	BDBM255370 (US9481682, 121) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	0.580	n/a	n/a	n/a	n/a	n/a	n/a
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Tyrosine-protein kinase FRK (Human)	BDBM255370 (US9481682, 121) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	530	n/a	n/a	n/a	n/a	n/a	n/a
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Tyrosine-protein kinase Fgr (Human)	BDBM255370 (US9481682, 121) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	263	n/a	n/a	n/a	n/a	n/a	n/a
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Receptor tyrosine-protein kinase erbB-4 (Human)	BDBM255370 (US9481682, 121) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	3.30E+3	n/a	n/a	n/a	n/a	n/a	n/a
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Tyrosine-protein kinase CSK (Human)	BDBM255370 (US9481682, 121) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	717	n/a	n/a	n/a	n/a	n/a	n/a
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Cytoplasmic tyrosine-protein kinase BMX (Human)	BDBM255370 (US9481682, 121) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	64	n/a	n/a	n/a	n/a	n/a	n/a
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Tyrosine-protein kinase Blk (Human)	BDBM255370 (US9481682, 121) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	309	n/a	n/a	n/a	n/a	n/a	n/a
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Tyrosine-protein kinase BTK (Human)	BDBM255370 (US9481682, 121) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	494	n/a	n/a	n/a	n/a	n/a	n/a
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					More data for this Ligand-Target Pair
Tyrosine-protein kinase BTK (Human)	BDBM255370 (US9481682, 121) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	12	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Tyrosine-protein kinase BTK (Human)	BDBM255370 (US9481682, 121) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	0.580	n/a	n/a	n/a	n/a	n/a	n/a
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