BDBM260253 US9522914, B-06

SMILES COc1cc(ccc1F)-c1nc(nn1CC(=O)NC(C)C)-c1ccc(CCN2C3CCC2COC3)cn1

InChI Key InChIKey=ZVWPUDSCBKVVLT-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 260253   

TargetVasopressin V1b receptor(Homo sapiens (Human))
Taisho Pharmaceutical

US Patent
LigandPNGBDBM260253(US9522914, B-06)
Affinity DataIC50:  3.30nMpH: 7.4 T: 2°CAssay Description:Human V1b receptor was transiently expressed in 293FT cells (Invitrogen). The cells were collected and then homogenated in a 15 mmol/L tris-hydrochlo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetVasopressin V1b receptor(Homo sapiens (Human))
Taisho Pharmaceutical

US Patent
LigandPNGBDBM260253(US9522914, B-06)
Affinity DataIC50:  3.30nMpH: 7.4 T: 2°CAssay Description:Human V1b receptor was transiently expressed in 293FT cells (Invitrogen). The cells were collected and then homogenated in a 15 mmol/L tris-hydrochlo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent