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BDBM26066 2-[(2-chloro-4-fluorophenyl)methyl]-3-(4-fluorophenyl)-7-(trifluoromethyl)-2H-indazole::JMC517161 Compound 12::US10543183, Compound LXR-623::US10669296, Compound LXR-623::US10945978, Compound 3::WAY-252623

SMILES: Fc1ccc(cc1)-c1n(Cc2ccc(F)cc2Cl)nc2c(cccc12)C(F)(F)F

InChI Key: InChIKey=KYWWJENKIMRJBI-UHFFFAOYSA-N

Data: 2 KI  2 IC50  14 EC50

Find this compound or compounds like it in BindingDB or PDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 16 hits for monomerid = 26066   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kcal/mole
IC50
nM
Kd
nM
EC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Oxysterols receptor LXR-beta [154-461]


(Human)
BDBM26066
PNG
(JMC517161 Compound 12 | 2-[(2-chloro-4-fluoropheny...)
GoogleScholar
UniChem
n/an/a 24n/a 3.67E+3n/an/a7.44


TBA



Citation and Details
More data for this
Ligand-Target Pair
Oxysterols receptor LXR-alpha [197-447]


(Human)
BDBM26066
PNG
(JMC517161 Compound 12 | 2-[(2-chloro-4-fluoropheny...)
GoogleScholar
UniChem
n/an/a 179n/a 6.66E+3n/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Oxysterols receptor LXR-alpha


(Human)
BDBM26066
PNG
(JMC517161 Compound 12 | 2-[(2-chloro-4-fluoropheny...)
GoogleScholar
UniChem
n/an/an/an/a 179n/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Oxysterols receptor LXR-beta


(Human)
BDBM26066
PNG
(JMC517161 Compound 12 | 2-[(2-chloro-4-fluoropheny...)
GoogleScholar
UniChem
n/an/an/an/a 24n/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Oxysterols receptor LXR-alpha


(Human)
BDBM26066
PNG
(JMC517161 Compound 12 | 2-[(2-chloro-4-fluoropheny...)
GoogleScholar
UniChem
n/an/an/an/a 179n/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Oxysterols receptor LXR-beta


(Human)
BDBM26066
PNG
(JMC517161 Compound 12 | 2-[(2-chloro-4-fluoropheny...)
GoogleScholar
UniChem
n/an/an/an/a 24n/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Oxysterols receptor LXR-alpha


(Human)
BDBM26066
PNG
(JMC517161 Compound 12 | 2-[(2-chloro-4-fluoropheny...)
GoogleScholar
UniChem
n/an/an/an/a 179n/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Oxysterols receptor LXR-beta


(Human)
BDBM26066
PNG
(JMC517161 Compound 12 | 2-[(2-chloro-4-fluoropheny...)
GoogleScholar
UniChem
n/an/an/an/a 24n/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Oxysterols receptor LXR-beta


(Human)
BDBM26066
PNG
(JMC517161 Compound 12 | 2-[(2-chloro-4-fluoropheny...)
GoogleScholar
UniChem
n/an/an/an/a 900n/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Oxysterols receptor LXR-alpha


(Human)
BDBM26066
PNG
(JMC517161 Compound 12 | 2-[(2-chloro-4-fluoropheny...)
GoogleScholar
UniChem
n/an/an/an/a 1.44E+3n/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Oxysterols receptor LXR-alpha/Retinoic acid receptor RXR-alpha


(Human)
BDBM26066
PNG
(JMC517161 Compound 12 | 2-[(2-chloro-4-fluoropheny...)
GoogleScholar
UniChem
n/an/an/an/a 0.431n/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Oxysterols receptor LXR-beta/Retinoic acid receptor RXR-alpha


(Human)
BDBM26066
PNG
(JMC517161 Compound 12 | 2-[(2-chloro-4-fluoropheny...)
GoogleScholar
UniChem
n/an/an/an/a 0.212n/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Oxysterols receptor LXR-beta


(Human)
BDBM26066
PNG
(JMC517161 Compound 12 | 2-[(2-chloro-4-fluoropheny...)
GoogleScholar
UniChem
n/an/an/an/a 3.67E+3n/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Oxysterols receptor LXR-alpha


(Human)
BDBM26066
PNG
(JMC517161 Compound 12 | 2-[(2-chloro-4-fluoropheny...)
GoogleScholar
UniChem
n/an/an/an/a 6.66E+3n/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Oxysterols receptor LXR-beta


(Human)
BDBM26066
PNG
(JMC517161 Compound 12 | 2-[(2-chloro-4-fluoropheny...)
GoogleScholar
UniChem
14n/an/an/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Oxysterols receptor LXR-beta


(Human)
BDBM26066
PNG
(JMC517161 Compound 12 | 2-[(2-chloro-4-fluoropheny...)
GoogleScholar
UniChem
14n/an/an/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair