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BDBM26145 2,4-dianilino pyrimidine, 2::3-({4-[(5-hydroxy-2-methylphenyl)amino]pyrimidin-2-yl}amino)benzamide::CHEMBL249097

SMILES: Cc1ccc(O)cc1Nc1ccnc(Nc2cccc(c2)C(N)=O)n1

InChI Key: InChIKey=SFCBIFOAGRZJNX-UHFFFAOYSA-N

Data: 1 IC50  18 Kd

Find this compound or compounds like it in BindingDB or PDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 19 hits for monomerid = 26145   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kcal/mole
IC50
nM
Kd
nM
EC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Protein-tyrosine kinase 6


(Human)
BDBM26145
PNG
(CHEMBL249097 | 3-({4-[(5-hydroxy-2-methylphenyl)am...)
GoogleScholar
UniChem
n/an/an/a 2n/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Atypical kinase COQ8B, mitochondrial


(Human)
BDBM26145
PNG
(CHEMBL249097 | 3-({4-[(5-hydroxy-2-methylphenyl)am...)
GoogleScholar
UniChem
n/an/an/a 129n/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Ephrin type-A receptor 2


(Human)
BDBM26145
PNG
(CHEMBL249097 | 3-({4-[(5-hydroxy-2-methylphenyl)am...)
GoogleScholar
UniChem
n/an/an/a 8n/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Ephrin type-B receptor 3


(Human)
BDBM26145
PNG
(CHEMBL249097 | 3-({4-[(5-hydroxy-2-methylphenyl)am...)
GoogleScholar
UniChem
n/an/an/a 81n/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Ephrin type-B receptor 2


(Human)
BDBM26145
PNG
(CHEMBL249097 | 3-({4-[(5-hydroxy-2-methylphenyl)am...)
GoogleScholar
UniChem
n/an/an/a 7n/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Ephrin type-A receptor 4


(Human)
BDBM26145
PNG
(CHEMBL249097 | 3-({4-[(5-hydroxy-2-methylphenyl)am...)
GoogleScholar
UniChem
n/an/an/a 5n/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Ephrin type-A receptor 5


(Human)
BDBM26145
PNG
(CHEMBL249097 | 3-({4-[(5-hydroxy-2-methylphenyl)am...)
GoogleScholar
UniChem
n/an/an/a 3n/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Ephrin type-A receptor 3


(Human)
BDBM26145
PNG
(CHEMBL249097 | 3-({4-[(5-hydroxy-2-methylphenyl)am...)
GoogleScholar
UniChem
n/an/an/a 0.100n/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Tyrosine-protein kinase receptor TYRO3


(Human)
BDBM26145
PNG
(CHEMBL249097 | 3-({4-[(5-hydroxy-2-methylphenyl)am...)
GoogleScholar
UniChem
n/an/an/a 264n/an/an/an/an/a


TBA



Citation and Details
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Ligand-Target Pair
Tyrosine-protein kinase CSK


(Human)
BDBM26145
PNG
(CHEMBL249097 | 3-({4-[(5-hydroxy-2-methylphenyl)am...)
GoogleScholar
UniChem
n/an/an/a 28n/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Proto-oncogene tyrosine-protein kinase LCK


(Mouse)
BDBM26145
PNG
(CHEMBL249097 | 3-({4-[(5-hydroxy-2-methylphenyl)am...)
GoogleScholar
UniChem
n/an/a 13n/an/an/an/a7.422


TBA



Citation and Details
More data for this
Ligand-Target Pair
Tyrosine-protein kinase Fgr


(Human)
BDBM26145
PNG
(CHEMBL249097 | 3-({4-[(5-hydroxy-2-methylphenyl)am...)
GoogleScholar
UniChem
n/an/an/a 0.300n/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Tyrosine-protein kinase Fyn


(Human)
BDBM26145
PNG
(CHEMBL249097 | 3-({4-[(5-hydroxy-2-methylphenyl)am...)
GoogleScholar
UniChem
n/an/an/a 0.400n/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Tyrosine-protein kinase Yes


(Human)
BDBM26145
PNG
(CHEMBL249097 | 3-({4-[(5-hydroxy-2-methylphenyl)am...)
GoogleScholar
UniChem
n/an/an/a 1n/an/an/an/an/a


TBA



Citation and Details
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Ligand-Target Pair
Tyrosine-protein kinase Blk


(Human)
BDBM26145
PNG
(CHEMBL249097 | 3-({4-[(5-hydroxy-2-methylphenyl)am...)
GoogleScholar
UniChem
n/an/an/a 1n/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Tyrosine-protein kinase TXK


(Human)
BDBM26145
PNG
(CHEMBL249097 | 3-({4-[(5-hydroxy-2-methylphenyl)am...)
GoogleScholar
UniChem
n/an/an/a 10n/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Cytoplasmic tyrosine-protein kinase BMX


(Human)
BDBM26145
PNG
(CHEMBL249097 | 3-({4-[(5-hydroxy-2-methylphenyl)am...)
GoogleScholar
UniChem
n/an/an/a 36n/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Ephrin type-A receptor 6


(Human)
BDBM26145
PNG
(CHEMBL249097 | 3-({4-[(5-hydroxy-2-methylphenyl)am...)
GoogleScholar
UniChem
n/an/an/a 20n/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Ephrin type-A receptor 1


(Human)
BDBM26145
PNG
(CHEMBL249097 | 3-({4-[(5-hydroxy-2-methylphenyl)am...)
GoogleScholar
UniChem
n/an/an/a 5n/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair