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BDBM261563 US9708270, 58

SMILES: Cc1ccc(C)c(c1)N1CCC2(CCC(CC(O)=O)CC2)CC1

InChI Key: InChIKey=MYXOTTPDDPJIOG-UHFFFAOYSA-N

Data: 1 EC50

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 261563   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kcal/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
G-protein coupled receptor 120


(Homo sapiens (Human))
BDBM261563
PNG
(US9708270, 58)
Show SMILES Cc1ccc(C)c(c1)N1CCC2(CCC(CC(O)=O)CC2)CC1
Show InChI InChI=1S/C20H29NO2/c1-15-3-4-16(2)18(13-15)21-11-9-20(10-12-21)7-5-17(6-8-20)14-19(22)23/h3-4,13,17H,5-12,14H2,1-2H3,(H,22,23)
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KEGG

UniProtKB/SwissProt

GoogleScholar
PC cid
PC sid
UniChem
US Patent
n/an/an/an/a 1.44E+3n/an/an/an/a



Merck Sharp & Dohme Corp

US Patent


Assay Description
On the day before the measurement day, CHO cells expressing human GPR120 were plated at 10000 cells per well in a 384-well black plate (#3702, Cornin...


US Patent US9708270 (2017)


BindingDB Entry DOI: 10.7270/Q24B33B5
More data for this
Ligand-Target Pair