BDBM26350 (S)-1-(2-oxo-1-(2-oxo-2-(pyrrolidin-1-yl)ethyl)azepan-3-yl)-3-m-tolylthiourea::1-(3-methylphenyl)-3-[(3S)-2-oxo-1-(2-oxo-2-pyrrolidin-1-ylethyl)azepan-3-yl]thiourea::3-(3-methylphenyl)-1-[(3S)-2-oxo-1-[2-oxo-2-(pyrrolidin-1-yl)ethyl]azepan-3-yl]thiourea::3-methylphenyl compound, 1::BMCL196882 Compound 1::CHEMBL198694
SMILES Cc1cccc(NC(=S)N[C@H]2CCCCN(CC(=O)N3CCCC3)C2=O)c1
InChI Key InChIKey=ROBFJTHBLVFFRU-KRWDZBQOSA-N
Data 5 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 5 hits for monomerid = 26350
Affinity DataIC50: 110nMpH: 7.4 T: 2°CAssay Description:Time-dependent optical density change was followed at 405 nm using a kinetic microplate reader at room temperature. Enzyme activity in the presence o...More data for this Ligand-Target Pair
Affinity DataIC50: 110nMpH: 7.4 T: 2°CAssay Description:Time-dependent optical density change was followed at 405 nm using a kinetic microplate reader at room temperature. Enzyme activity in the presence o...More data for this Ligand-Target Pair
Affinity DataIC50: 110nMAssay Description:Inhibition of factor 10aMore data for this Ligand-Target Pair
Affinity DataIC50: 110nMAssay Description:Inhibition of human factor 10a-mediated cleavage of synthetic substrate S-2222More data for this Ligand-Target Pair
Affinity DataIC50: 110nMAssay Description:Inhibitory activity against human FXaMore data for this Ligand-Target Pair