BDBM267010 US9718808, 139

SMILES CN(C)C(=O)CN(Cc1ccc(nc1)-n1cnnn1)[C@H]1CC[C@]2(CCN(C3=C(C)C(=O)OC3)C2=O)CC1

InChI Key InChIKey=UJGCILCVESUJIL-KJDSRRNHSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 267010   

TargetATP-sensitive inward rectifier potassium channel 1(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM267010(US9718808, 139)
Affinity DataIC50:  120nMAssay Description:A Thallium Flux Assay was performed on each of the final product compounds of the Examples. This assay has been described previously; see, e.g., PCT ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent