BDBM268510 N-(6-cyclopropyl-7-(spiro[5.5]undecan-3-yloxy)-[1,2,4]triazolo-[4,3-a]pyridin-3-yl)cyclopropanesulfonamide::US9550775, 35::US9550775, 90

SMILES O=S(=O)(Nc1nnc2cc(OC3CCC4(CCCCC4)CC3)c(cn12)C1CC1)C1CC1

InChI Key InChIKey=GDYONBVASIDQMC-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 268510   

TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM268510(N-(6-cyclopropyl-7-(spiro[5.5]undecan-3-yloxy)-[1,...)
Affinity DataIC50:  51nMpH: 7.2Assay Description:The following patch voltage clamp electrophysiology studies were performed on representative compounds of the invention using human embryonic kidney ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM268510(N-(6-cyclopropyl-7-(spiro[5.5]undecan-3-yloxy)-[1,...)
Affinity DataIC50:  51.3nMpH: 7.2Assay Description:The following patch voltage clamp electrophysiology studies were performed on representative compounds of the invention using human embryonic kidney ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent