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BDBM26890 8-(diphenylmethyl)-3-ethyl-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one::spiropiperidine analogue, 11

SMILES: CCN1CN(c2ccccc2)C2(CCN(CC2)C(c2ccccc2)c2ccccc2)C1=O

InChI Key: InChIKey=AJCMEBINTIHGEB-UHFFFAOYSA-N

Data: 4 KI

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 26890
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Nociceptin receptor (Human)	BDBM26890 (8-(diphenylmethyl)-3-ethyl-1-phenyl-1,3,8-triazasp...) Show SMILES Show InChI	GoogleScholar	UniChem		84	-9.55	n/a	n/a	n/a	n/a	n/a	7.4	22
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Kappa-type opioid receptor (Human)	BDBM26890 (8-(diphenylmethyl)-3-ethyl-1-phenyl-1,3,8-triazasp...) Show SMILES Show InChI	GoogleScholar	UniChem		506	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Mu-type opioid receptor (Human)	BDBM26890 (8-(diphenylmethyl)-3-ethyl-1-phenyl-1,3,8-triazasp...) Show SMILES Show InChI	GoogleScholar	UniChem		2.28E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Delta-type opioid receptor (Human)	BDBM26890 (8-(diphenylmethyl)-3-ethyl-1-phenyl-1,3,8-triazasp...) Show SMILES Show InChI	GoogleScholar	UniChem		2.32E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair