BDBM27165 1H-indol-1-yl tertiary amine, 9::methyl 3-[3-({[2-chloro-3-(trifluoromethyl)phenyl]methyl}(2,2-diphenylethyl)amino)propoxy]-1,2-oxazole-5-carboxylate

SMILES COC(=O)c1cc(OCCCN(CC(c2ccccc2)c2ccccc2)Cc2cccc(c2Cl)C(F)(F)F)no1

InChI Key InChIKey=UMYHRDJPCVNPPU-UHFFFAOYSA-N

Data  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 27165   

TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Gsk

LigandPNGBDBM27165(1H-indol-1-yl tertiary amine, 9 | methyl 3-[3-({[2...)
Affinity DataEC50:  26nMpH: 7.5 T: 2°CAssay Description:The LXR LiSA measures the ligand-dependent recruitment of a 25 amino acid fragment of the steroid receptor coactivator 1 (SRC1) to the ligand-binding...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Gsk

LigandPNGBDBM27165(1H-indol-1-yl tertiary amine, 9 | methyl 3-[3-({[2...)
Affinity DataEC50:  63nMpH: 7.5 T: 2°CAssay Description:The LXR LiSA measures the ligand-dependent recruitment of a 25 amino acid fragment of the steroid receptor coactivator 1 (SRC1) to the ligand-binding...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed