BDBM27213 4-[3-(4-cyclopropanecarbonylphenoxy)propyl]-1H-imidazole::CHEMBL14638::CHEMBL1795025::Ciproxifan

SMILES: O=C(C1CC1)c1ccc(OCCCc2cnc[nH]2)cc1

InChI Key: InChIKey=ACQBHJXEAYTHCY-UHFFFAOYSA-N

Data: 51 KI  1 IC50

Find this compound or compounds like it in BindingDB or PDB:

Substructure Similarity at least:  must be >=0.5 Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 52 hits for monomerid = 27213   

Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50 nM	koff s-1	kon M-1s-1	pH	Temp °C
Histamine N-methyltransferase (Rat)	BDBM27213 (CHEMBL1795025 | 4-[3-(4-cyclopropanecarbonylphenox...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	9.00E+3	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Hrh3 protein (Rat)	BDBM27213 (CHEMBL1795025 | 4-[3-(4-cyclopropanecarbonylphenox...) Show SMILES Show InChI	GoogleScholar	UniChem		0.427	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Histamine H3 receptor (Rat)	BDBM27213 (CHEMBL1795025 | 4-[3-(4-cyclopropanecarbonylphenox...) Show SMILES Show InChI	GoogleScholar	UniChem		0.490	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Histamine H3 receptor (Rat)	BDBM27213 (CHEMBL1795025 | 4-[3-(4-cyclopropanecarbonylphenox...) Show SMILES Show InChI	GoogleScholar	UniChem		0.490	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Histamine H3 receptor (Rat)	BDBM27213 (CHEMBL1795025 | 4-[3-(4-cyclopropanecarbonylphenox...) Show SMILES Show InChI	GoogleScholar	UniChem		0.490	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Histamine H3 receptor (Rat)	BDBM27213 (CHEMBL1795025 | 4-[3-(4-cyclopropanecarbonylphenox...) Show SMILES Show InChI	GoogleScholar	UniChem		0.490	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Hrh3 protein (Rat)	BDBM27213 (CHEMBL1795025 | 4-[3-(4-cyclopropanecarbonylphenox...) Show SMILES Show InChI	GoogleScholar	UniChem		0.510	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Histamine H3 receptor (Rat)	BDBM27213 (CHEMBL1795025 | 4-[3-(4-cyclopropanecarbonylphenox...) Show SMILES Show InChI	GoogleScholar	UniChem		0.510	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Hrh3 protein (Rat)	BDBM27213 (CHEMBL1795025 | 4-[3-(4-cyclopropanecarbonylphenox...) Show SMILES Show InChI	GoogleScholar	UniChem		0.510	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Histamine H3 receptor (Rat)	BDBM27213 (CHEMBL1795025 | 4-[3-(4-cyclopropanecarbonylphenox...) Show SMILES Show InChI	GoogleScholar	UniChem		0.630	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Hrh3 protein (Rat)	BDBM27213 (CHEMBL1795025 | 4-[3-(4-cyclopropanecarbonylphenox...) Show SMILES Show InChI	GoogleScholar	UniChem		0.630	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Hrh3 protein (Rat)	BDBM27213 (CHEMBL1795025 | 4-[3-(4-cyclopropanecarbonylphenox...) Show SMILES Show InChI	GoogleScholar	UniChem		0.630	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Hrh3 protein (Rat)	BDBM27213 (CHEMBL1795025 | 4-[3-(4-cyclopropanecarbonylphenox...) Show SMILES Show InChI	GoogleScholar	UniChem		0.654	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Histamine H3 receptor (Guinea pig)	BDBM27213 (CHEMBL1795025 | 4-[3-(4-cyclopropanecarbonylphenox...) Show SMILES Show InChI	GoogleScholar	UniChem		1.74	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Histamine H3 receptor (Guinea pig)	BDBM27213 (CHEMBL1795025 | 4-[3-(4-cyclopropanecarbonylphenox...) Show SMILES Show InChI	GoogleScholar	UniChem		1.74	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Histamine H3 receptor (Rat)	BDBM27213 (CHEMBL1795025 | 4-[3-(4-cyclopropanecarbonylphenox...) Show SMILES Show InChI	GoogleScholar	UniChem		3.90	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Histamine receptor H3 (Dog)	BDBM27213 (CHEMBL1795025 | 4-[3-(4-cyclopropanecarbonylphenox...) Show SMILES Show InChI	GoogleScholar	UniChem		5.75	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Histamine receptor H3 (Dog)	BDBM27213 (CHEMBL1795025 | 4-[3-(4-cyclopropanecarbonylphenox...) Show SMILES Show InChI	GoogleScholar	UniChem		5.75	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Alpha-2A adrenergic receptor (Human)	BDBM27213 (CHEMBL1795025 | 4-[3-(4-cyclopropanecarbonylphenox...) Show SMILES Show InChI	GoogleScholar	UniChem		42.7	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Histamine H3 receptor (Human)	BDBM27213 (CHEMBL1795025 | 4-[3-(4-cyclopropanecarbonylphenox...) Show SMILES Show InChI	GoogleScholar	UniChem		46	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Histamine H3 receptor (Human)	BDBM27213 (CHEMBL1795025 | 4-[3-(4-cyclopropanecarbonylphenox...) Show SMILES Show InChI	GoogleScholar	UniChem		46	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Histamine H3 receptor (Human)	BDBM27213 (CHEMBL1795025 | 4-[3-(4-cyclopropanecarbonylphenox...) Show SMILES Show InChI	GoogleScholar	UniChem		46	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Histamine H3 receptor (Human)	BDBM27213 (CHEMBL1795025 | 4-[3-(4-cyclopropanecarbonylphenox...) Show SMILES Show InChI	GoogleScholar	UniChem		46	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Histamine H3 receptor (Human)	BDBM27213 (CHEMBL1795025 | 4-[3-(4-cyclopropanecarbonylphenox...) Show SMILES Show InChI	GoogleScholar	UniChem		46	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Histamine H3 receptor (Human)	BDBM27213 (CHEMBL1795025 | 4-[3-(4-cyclopropanecarbonylphenox...) Show SMILES Show InChI	GoogleScholar	UniChem		62.5	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Histamine H3 receptor (Human)	BDBM27213 (CHEMBL1795025 | 4-[3-(4-cyclopropanecarbonylphenox...) Show SMILES Show InChI	GoogleScholar	UniChem		63	-9.82	n/a	n/a	n/a	n/a	n/a	7.4	25
TBA									Citation and Details
					More data for this Ligand-Target Pair
Histamine H3 receptor (Human)	BDBM27213 (CHEMBL1795025 | 4-[3-(4-cyclopropanecarbonylphenox...) Show SMILES Show InChI	GoogleScholar	UniChem		63	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Histamine H3 receptor (Human)	BDBM27213 (CHEMBL1795025 | 4-[3-(4-cyclopropanecarbonylphenox...) Show SMILES Show InChI	GoogleScholar	UniChem		63	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Histamine H3 receptor (Human)	BDBM27213 (CHEMBL1795025 | 4-[3-(4-cyclopropanecarbonylphenox...) Show SMILES Show InChI	GoogleScholar	UniChem		63.1	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Alpha-2C adrenergic receptor (Human)	BDBM27213 (CHEMBL1795025 | 4-[3-(4-cyclopropanecarbonylphenox...) Show SMILES Show InChI	GoogleScholar	UniChem		63.1	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Histamine H3 receptor (Human)	BDBM27213 (CHEMBL1795025 | 4-[3-(4-cyclopropanecarbonylphenox...) Show SMILES Show InChI	GoogleScholar	UniChem		63.1	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Histamine H3 receptor (Human)	BDBM27213 (CHEMBL1795025 | 4-[3-(4-cyclopropanecarbonylphenox...) Show SMILES Show InChI	GoogleScholar	UniChem		89.1	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Histamine H3 receptor (Human)	BDBM27213 (CHEMBL1795025 | 4-[3-(4-cyclopropanecarbonylphenox...) Show SMILES Show InChI	GoogleScholar	UniChem		89.1	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Histamine H3 receptor (Human)	BDBM27213 (CHEMBL1795025 | 4-[3-(4-cyclopropanecarbonylphenox...) Show SMILES Show InChI	GoogleScholar	UniChem		89.4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Histamine H3 receptor (Human)	BDBM27213 (CHEMBL1795025 | 4-[3-(4-cyclopropanecarbonylphenox...) Show SMILES Show InChI	GoogleScholar	UniChem		94	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Histamine H3 receptor (Human)	BDBM27213 (CHEMBL1795025 | 4-[3-(4-cyclopropanecarbonylphenox...) Show SMILES Show InChI	GoogleScholar	UniChem		94	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
5-hydroxytryptamine receptor 3A (Rat)	BDBM27213 (CHEMBL1795025 | 4-[3-(4-cyclopropanecarbonylphenox...) Show SMILES Show InChI	GoogleScholar	UniChem		302	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Histamine H4 receptor (Human)	BDBM27213 (CHEMBL1795025 | 4-[3-(4-cyclopropanecarbonylphenox...) Show SMILES Show InChI	GoogleScholar	UniChem		612	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Histamine H4 receptor (Human)	BDBM27213 (CHEMBL1795025 | 4-[3-(4-cyclopropanecarbonylphenox...) Show SMILES Show InChI	GoogleScholar	UniChem		612	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Histamine H4 receptor (Human)	BDBM27213 (CHEMBL1795025 | 4-[3-(4-cyclopropanecarbonylphenox...) Show SMILES Show InChI	GoogleScholar	UniChem		1.86E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Histamine H4 receptor (Human)	BDBM27213 (CHEMBL1795025 | 4-[3-(4-cyclopropanecarbonylphenox...) Show SMILES Show InChI	GoogleScholar	UniChem		1.86E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Histamine H4 receptor (Human)	BDBM27213 (CHEMBL1795025 | 4-[3-(4-cyclopropanecarbonylphenox...) Show SMILES Show InChI	GoogleScholar	UniChem		1.86E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Histamine H4 receptor (Human)	BDBM27213 (CHEMBL1795025 | 4-[3-(4-cyclopropanecarbonylphenox...) Show SMILES Show InChI	GoogleScholar	UniChem		1.88E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Histamine H1 receptor (Human)	BDBM27213 (CHEMBL1795025 | 4-[3-(4-cyclopropanecarbonylphenox...) Show SMILES Show InChI	GoogleScholar	UniChem		>2.51E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
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Histamine H2 receptor (Human)	BDBM27213 (CHEMBL1795025 | 4-[3-(4-cyclopropanecarbonylphenox...) Show SMILES Show InChI	GoogleScholar	UniChem		>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Histamine H1 receptor (Human)	BDBM27213 (CHEMBL1795025 | 4-[3-(4-cyclopropanecarbonylphenox...) Show SMILES Show InChI	GoogleScholar	UniChem		>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Histamine H2 receptor (Human)	BDBM27213 (CHEMBL1795025 | 4-[3-(4-cyclopropanecarbonylphenox...) Show SMILES Show InChI	GoogleScholar	UniChem		>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Histamine H1 receptor (Human)	BDBM27213 (CHEMBL1795025 | 4-[3-(4-cyclopropanecarbonylphenox...) Show SMILES Show InChI	GoogleScholar	UniChem		>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Histamine H2 receptor (Human)	BDBM27213 (CHEMBL1795025 | 4-[3-(4-cyclopropanecarbonylphenox...) Show SMILES Show InChI	GoogleScholar	UniChem		>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
Histamine H1 receptor (Human)	BDBM27213 (CHEMBL1795025 | 4-[3-(4-cyclopropanecarbonylphenox...) Show SMILES Show InChI	GoogleScholar	UniChem		>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair