BDBM27217 (2R)-2-{[4-(benzylamino)-8-(propan-2-yl)pyrazolo[1,5-a][1,3,5]triazin-2-yl]amino}butan-1-ol::GP0210::pyrazolo[1,5-a]-1,3,5-triazine, 7a

SMILES: CC[C@H](CO)Nc1nc(NCc2ccccc2)n2ncc(C(C)C)c2n1

InChI Key: InChIKey=SQUNOCMDMIQIQK-UHFFFAOYSA-N

Data: 15 IC50

Find this compound or compounds like it in BindingDB or PDB:

Substructure Similarity at least:  must be >=0.5 Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 15 hits for monomerid = 27217   

Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50 nM	koff s-1	kon M-1s-1	pH	Temp °C
Cyclin-dependent kinase/G2/mitotic-specific cyclin- 1 (Human)	BDBM27217 (GP0210 | (2R)-2-{[4-(benzylamino)-8-(propan-2-yl)p...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	73	n/a	n/a	n/a	n/a	7.5	30
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Cyclin-A2/Cyclin-dependent kinase 2 (Human)	BDBM27217 (GP0210 | (2R)-2-{[4-(benzylamino)-8-(propan-2-yl)p...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	40	n/a	n/a	n/a	n/a	7.5	30
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Cyclin-dependent kinase 5 activator 1 [99-307] (Human)	BDBM27217 (GP0210 | (2R)-2-{[4-(benzylamino)-8-(propan-2-yl)p...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	70	n/a	n/a	n/a	n/a	7.5	30
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Cyclin-H/Cyclin-dependent kinase 7 (Human)	BDBM27217 (GP0210 | (2R)-2-{[4-(benzylamino)-8-(propan-2-yl)p...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	500	n/a	n/a	n/a	n/a	7.5	30
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Cyclin-T1/Cyclin-dependent kinase 9 (Human)	BDBM27217 (GP0210 | (2R)-2-{[4-(benzylamino)-8-(propan-2-yl)p...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	43	n/a	n/a	n/a	n/a	7.5	30
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Dual specificity tyrosine-phosphorylation-regulated kinase 1A (Rat)	BDBM27217 (GP0210 | (2R)-2-{[4-(benzylamino)-8-(propan-2-yl)p...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	1.30E+3	n/a	n/a	n/a	n/a	n/a	n/a
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Cyclin-dependent kinase 5 activator 1 (Human)	BDBM27217 (GP0210 | (2R)-2-{[4-(benzylamino)-8-(propan-2-yl)p...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	43	n/a	n/a	n/a	n/a	n/a	n/a
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Cyclin-A2/Cyclin-dependent kinase 2 (Human)	BDBM27217 (GP0210 | (2R)-2-{[4-(benzylamino)-8-(propan-2-yl)p...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	43	n/a	n/a	n/a	n/a	n/a	n/a
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Cyclin-H/Cyclin-dependent kinase 7 (Human)	BDBM27217 (GP0210 | (2R)-2-{[4-(benzylamino)-8-(propan-2-yl)p...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	43	n/a	n/a	n/a	n/a	n/a	n/a
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Cyclin-T1/Cyclin-dependent kinase 9 (Human)	BDBM27217 (GP0210 | (2R)-2-{[4-(benzylamino)-8-(propan-2-yl)p...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	43	n/a	n/a	n/a	n/a	n/a	n/a
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Cyclin-dependent kinase 2/G1/S-specific cyclin-E1 (Human)	BDBM27217 (GP0210 | (2R)-2-{[4-(benzylamino)-8-(propan-2-yl)p...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	43	n/a	n/a	n/a	n/a	n/a	n/a
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Cyclin-A2/Cyclin-dependent kinase 2 (Human)	BDBM27217 (GP0210 | (2R)-2-{[4-(benzylamino)-8-(propan-2-yl)p...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	40	n/a	n/a	n/a	n/a	n/a	n/a
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					More data for this Ligand-Target Pair
Cyclin-dependent kinase 2/G1/S-specific cyclin-E1 (Human)	BDBM27217 (GP0210 | (2R)-2-{[4-(benzylamino)-8-(propan-2-yl)p...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	26	n/a	n/a	n/a	n/a	n/a	n/a
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Cyclin-dependent kinase 5 activator 1 (Human)	BDBM27217 (GP0210 | (2R)-2-{[4-(benzylamino)-8-(propan-2-yl)p...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	70	n/a	n/a	n/a	n/a	n/a	n/a
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					More data for this Ligand-Target Pair
Cyclin-T1/Cyclin-dependent kinase 9 (Human)	BDBM27217 (GP0210 | (2R)-2-{[4-(benzylamino)-8-(propan-2-yl)p...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	43	n/a	n/a	n/a	n/a	n/a	n/a
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					More data for this Ligand-Target Pair