BDBM283058 6-(1-(2,2-difluoroethyl)-4-(3- (trifluoromethoxy)phenyl)-1H-imidazol-5- yl)imidazo[1,2-b]pyridazine-3-carbonitrile::US10287295, Example 259'::US11352360, Example 259'::US9884868, Example 259'
SMILES FC(F)Cn1cnc(c1-c1ccc2ncc(C#N)n2n1)-c1cccc(OC(F)(F)F)c1
InChI Key InChIKey=KTYXJOHTTOOMEL-UHFFFAOYSA-N
Data 6 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 6 hits for monomerid = 283058
Affinity DataIC50: 1nMpH: 7.4 T: 2°CAssay Description:Assays for the compounds reported below were conducted in 1536-well plates and 2 mL reactions are prepared from addition of HIS-TGF-βR1 T204D or...More data for this Ligand-Target Pair
Affinity DataIC50: >1.50E+4nMAssay Description:Assays for the compounds reported below were conducted in 1536-well plates and 2 mL reactions are prepared from addition of HIS-TGF-βR1 T204D or...More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Assays for the compounds reported below were conducted in 1536-well plates and 2 mL reactions are prepared from addition of HIS-TGF-βR1 T204D or...More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Assays for the compounds reported below were conducted in 1536-well plates and 2 mL reactions are prepared from addition of HIS-TGF-βR1 T204D or...More data for this Ligand-Target Pair