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BDBM29075 PF-514273

SMILES: CC(F)(F)CN1CCOc2c(nn(c2-c2ccc(Cl)cc2)-c2ccccc2Cl)C1=O

InChI Key: InChIKey=FJMQJSUOOGOWBD-UHFFFAOYSA-N

Data: 5 KI 1 EC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 5 hits for monomerid = 29075
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Cannabinoid receptor 1 (Human)	BDBM29075 (PF-514273) Show SMILES Show InChI	GoogleScholar	UniChem		0.820	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Cannabinoid receptor 1 (Human)	BDBM29075 (PF-514273) Show SMILES Show InChI	GoogleScholar	UniChem		1	-12.5	n/a	n/a	0.820	n/a	n/a	7.4	30
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Cannabinoid receptor 1 (Human)	BDBM29075 (PF-514273) Show SMILES Show InChI	GoogleScholar	UniChem		1	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Cannabinoid receptor 2 (Human)	BDBM29075 (PF-514273) Show SMILES Show InChI	GoogleScholar	UniChem		>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Cannabinoid receptor 2 (Human)	BDBM29075 (PF-514273) Show SMILES Show InChI	GoogleScholar	UniChem		>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair