BDBM297503 N-{4-[4-(2-azetidin-1-yl-phenyl)- piperidin-1-yl]-2-cyclopropyl- quinazolin-6-yl}-N,N',N'- trimethyl-ethane-1,2-diamine::US10118902, Example 5::US10584103, Example 5

SMILES CN(C)CCN(C)c1ccc2nc(nc(N3CCC(CC3)c3ccccc3N3CCC3)c2c1)C1CC1

InChI Key InChIKey=BNRSTXNKEMTKFL-UHFFFAOYSA-N

Data  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 297503   

TargetNeurotensin receptor type 1(Homo sapiens (Human))
Sanford Burnham Prebys Medical Discovery Institute

US Patent
LigandPNGBDBM297503(N-{4-[4-(2-azetidin-1-yl-phenyl)- piperidin-1-yl]-...)
Affinity DataEC50:  6.00E+3nMAssay Description:NTSR1 (NTR1) CHO cells are plated in 20 μL of assay media containing Ham's F12 supplemented with 10% fetal bovine serum and 0.4 mg/mL G418 a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetNeurotensin receptor type 1(Homo sapiens (Human))
Sanford Burnham Prebys Medical Discovery Institute

US Patent
LigandPNGBDBM297503(N-{4-[4-(2-azetidin-1-yl-phenyl)- piperidin-1-yl]-...)
Affinity DataEC50:  6.00E+3nMAssay Description:NTSR1 (NTR1) CHO cells are plated in 20 uL of assay media containing Ham's F12 supplemented with 10% fetal bovine serum and 0.4 mg/mL G418 at a c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent