BDBM301991 2-(4-(4-(5-Cyano-1H-indol-3-yl)butyl)piperazin-1-yl)-4-methylthiazole-5-carbonitrile::US9598401, Example 47
SMILES Cc1nc(sc1C#N)N1CCN(CCCCc2c[nH]c3ccc(cc23)C#N)CC1
InChI Key InChIKey=XGLGVMXPTXRAKN-UHFFFAOYSA-N
Data 2 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 301991
Affinity DataKi: 5nMAssay Description:Human HEK-293 cell homogenates (36 μg protein) were incubated at 22° C. for 60 minutes with 0.3 nM [3H]8-OH-DPAT (Perkin-Elmer) in the absence o...More data for this Ligand-Target Pair
Affinity DataKi: 130nMAssay Description:Cell membrane homogenates (24 μg protein) were incubated at 22° C. for 60 minutes with 0.3 nM [3H]methyl-spiperone in the absence or presence of...More data for this Ligand-Target Pair