BDBM305967 US10144742, Compound I-129

SMILES CS(=O)(=O)N1CCN(CC1)c1nc2cc(ccc2nc1-c1ccccc1)C(=O)NCCCn1ccnc1

InChI Key InChIKey=DYFXJTHSNLEHEE-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 305967   

TargetNicotinamide phosphoribosyltransferase(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM305967(US10144742, Compound I-129)
Affinity DataIC50:  300nMAssay Description:To measure the inhibition of NAMPT activity hNAMPT protein stock and anti 6His-Tb (Cisbio; Cat. No. 61HISTLB) is diluted to 3× final concentration wi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent