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BDBM310898 N,N-dimethyl-3-(6-methyl-7-oxo-1H-pyrrolo[2,3-c]pyridin-4-yl)benzamide::US10150767, Example 22

SMILES: CN1C=C(c2cc[nH]c2C1=O)c3cccc(c3)C(=O)N(C)C

InChI Key: InChIKey=YHMNROQTPUKNLA-UHFFFAOYSA-N

Data: 38 IC50

PDB links: 3 PDB IDs match this monomer.

Find this compound or compounds like it in BindingDB or PDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 38 hits for monomerid = 310898   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kcal/mole
IC50
nM
Kd
nM
EC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Transcription intermediary factor 1-alpha


(Human)
BDBM310898
PNG
(US10150767, Example 22 | N,N-dimethyl-3-(6-methyl-...)
GoogleScholar
UniChem
n/an/a 910n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Histone acetyltransferase p300


(Human)
BDBM310898
PNG
(US10150767, Example 22 | N,N-dimethyl-3-(6-methyl-...)
GoogleScholar
UniChem
n/an/a 270n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Bromodomain adjacent to zinc finger domain protein 2B


(Human)
BDBM310898
PNG
(US10150767, Example 22 | N,N-dimethyl-3-(6-methyl-...)
GoogleScholar
UniChem
n/an/a 3.60E+3n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Transcription activator BRG1


(Human)
BDBM310898
PNG
(US10150767, Example 22 | N,N-dimethyl-3-(6-methyl-...)
GoogleScholar
UniChem
n/an/a 9.00E+3n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Transcription initiation factor TFIID subunit 1


(Human)
BDBM310898
PNG
(US10150767, Example 22 | N,N-dimethyl-3-(6-methyl-...)
GoogleScholar
UniChem
n/an/a 59n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Transcription initiation factor TFIID subunit 1


(Human)
BDBM310898
PNG
(US10150767, Example 22 | N,N-dimethyl-3-(6-methyl-...)
GoogleScholar
UniChem
n/an/a 3.60E+3n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Bromodomain-containing protein 9


(Human)
BDBM310898
PNG
(US10150767, Example 22 | N,N-dimethyl-3-(6-methyl-...)
GoogleScholar
UniChem
n/an/a 230n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
CREB-binding protein


(Human)
BDBM310898
PNG
(US10150767, Example 22 | N,N-dimethyl-3-(6-methyl-...)
GoogleScholar
UniChem
n/an/a 560n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Bromodomain-containing protein 4


(Human)
BDBM310898
PNG
(US10150767, Example 22 | N,N-dimethyl-3-(6-methyl-...)
GoogleScholar
UniChem
n/an/a 65n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Bromodomain-containing protein 4


(Human)
BDBM310898
PNG
(US10150767, Example 22 | N,N-dimethyl-3-(6-methyl-...)
GoogleScholar
UniChem
n/an/a 92n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Bromodomain-containing protein 4


(Human)
BDBM310898
PNG
(US10150767, Example 22 | N,N-dimethyl-3-(6-methyl-...)
GoogleScholar
UniChem
n/an/a 92n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Protein polybromo-1


(Human)
BDBM310898
PNG
(US10150767, Example 22 | N,N-dimethyl-3-(6-methyl-...)
GoogleScholar
UniChem
n/an/a 7.60E+3n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Peregrin


(Human)
BDBM310898
PNG
(US10150767, Example 22 | N,N-dimethyl-3-(6-methyl-...)
GoogleScholar
UniChem
n/an/a 1.50E+3n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Peregrin


(Human)
BDBM310898
PNG
(US10150767, Example 22 | N,N-dimethyl-3-(6-methyl-...)
GoogleScholar
UniChem
n/an/a 1.50E+3n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Bromodomain adjacent to zinc finger domain protein 2A


(Human)
BDBM310898
PNG
(US10150767, Example 22 | N,N-dimethyl-3-(6-methyl-...)
GoogleScholar
UniChem
n/an/a 880n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Protein polybromo-1


(Human)
BDBM310898
PNG
(US10150767, Example 22 | N,N-dimethyl-3-(6-methyl-...)
GoogleScholar
UniChem
n/an/a 7.60E+3n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Chromatin remodeling regulator CECR2


(Human)
BDBM310898
PNG
(US10150767, Example 22 | N,N-dimethyl-3-(6-methyl-...)
GoogleScholar
UniChem
n/an/a 240n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Probable global transcription activator SNF2L2


(Human)
BDBM310898
PNG
(US10150767, Example 22 | N,N-dimethyl-3-(6-methyl-...)
GoogleScholar
UniChem
n/an/a 6.70E+3n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Probable global transcription activator SNF2L2


(Human)
BDBM310898
PNG
(US10150767, Example 22 | N,N-dimethyl-3-(6-methyl-...)
GoogleScholar
UniChem
n/an/a 6.70E+3n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Histone acetyltransferase p300


(Human)
BDBM310898
PNG
(US10150767, Example 22 | N,N-dimethyl-3-(6-methyl-...)
GoogleScholar
UniChem
n/an/a 270n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Transcription initiation factor TFIID subunit 1


(Human)
BDBM310898
PNG
(US10150767, Example 22 | N,N-dimethyl-3-(6-methyl-...)
GoogleScholar
UniChem
n/an/a 59n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Bromodomain-containing protein 4


(Human)
BDBM310898
PNG
(US10150767, Example 22 | N,N-dimethyl-3-(6-methyl-...)
GoogleScholar
UniChem
n/an/a 65n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Chromatin remodeling regulator CECR2


(Human)
BDBM310898
PNG
(US10150767, Example 22 | N,N-dimethyl-3-(6-methyl-...)
GoogleScholar
UniChem
n/an/a 240n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
CREB-binding protein


(Human)
BDBM310898
PNG
(US10150767, Example 22 | N,N-dimethyl-3-(6-methyl-...)
GoogleScholar
UniChem
n/an/a 560n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Bromodomain-containing protein 4


(Human)
BDBM310898
PNG
(US10150767, Example 22 | N,N-dimethyl-3-(6-methyl-...)
GoogleScholar
UniChem
n/an/a 92n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Transcription initiation factor TFIID subunit 1


(Human)
BDBM310898
PNG
(US10150767, Example 22 | N,N-dimethyl-3-(6-methyl-...)
GoogleScholar
UniChem
n/an/a 3.60E+3n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Bromodomain-containing protein 9


(Human)
BDBM310898
PNG
(US10150767, Example 22 | N,N-dimethyl-3-(6-methyl-...)
GoogleScholar
UniChem
n/an/a 230n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Bromodomain adjacent to zinc finger domain protein 2A


(Human)
BDBM310898
PNG
(US10150767, Example 22 | N,N-dimethyl-3-(6-methyl-...)
GoogleScholar
UniChem
n/an/a 880n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Transcription intermediary factor 1-alpha


(Human)
BDBM310898
PNG
(US10150767, Example 22 | N,N-dimethyl-3-(6-methyl-...)
GoogleScholar
UniChem
n/an/a 910n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Bromodomain-containing protein 9 [134-239]


(Human)
BDBM310898
PNG
(US10150767, Example 22 | N,N-dimethyl-3-(6-methyl-...)
GoogleScholar
UniChem
n/an/a 53n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Bromodomain adjacent to zinc finger domain protein 2B


(Human)
BDBM310898
PNG
(US10150767, Example 22 | N,N-dimethyl-3-(6-methyl-...)
GoogleScholar
UniChem
n/an/a 3.60E+3n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Transcription activator BRG1


(Human)
BDBM310898
PNG
(US10150767, Example 22 | N,N-dimethyl-3-(6-methyl-...)
GoogleScholar
UniChem
n/an/a 9.00E+3n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Chromatin remodeling regulator CECR2


(Human)
BDBM310898
PNG
(US10150767, Example 22 | N,N-dimethyl-3-(6-methyl-...)
GoogleScholar
UniChem
n/an/a 240n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Transcription initiation factor TFIID subunit 1


(Human)
BDBM310898
PNG
(US10150767, Example 22 | N,N-dimethyl-3-(6-methyl-...)
GoogleScholar
UniChem
n/an/a 59n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Transcription initiation factor TFIID subunit 1


(Human)
BDBM310898
PNG
(US10150767, Example 22 | N,N-dimethyl-3-(6-methyl-...)
GoogleScholar
UniChem
n/an/a 3.60E+3n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Bromodomain-containing protein 9


(Human)
BDBM310898
PNG
(US10150767, Example 22 | N,N-dimethyl-3-(6-methyl-...)
GoogleScholar
UniChem
n/an/a 230n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
CREB-binding protein


(Human)
BDBM310898
PNG
(US10150767, Example 22 | N,N-dimethyl-3-(6-methyl-...)
GoogleScholar
UniChem
n/an/a 560n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Bromodomain-containing protein 4


(Human)
BDBM310898
PNG
(US10150767, Example 22 | N,N-dimethyl-3-(6-methyl-...)
GoogleScholar
UniChem
n/an/a 65n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair