BDBM328072 5-(3-(4- cyanophenoxy)azetidine- 1-carbonyl)-N-(6-(4- fluorophenoxy)pyridin- 3-yl)picolinamide::US10377742, Compound 210::US9663496, Compound 210

SMILES Fc1ccc(Oc2ccc(NC(=O)c3ccc(cn3)C(=O)N3CC(C3)Oc3ccc(cc3)C#N)cn2)cc1

InChI Key InChIKey=JGBMPZMXPFSPDG-UHFFFAOYSA-N

Data  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 328072   

Target5'-AMP-activated protein kinase catalytic subunit alpha-2(Homo sapiens (Human))
Rigel Pharmaceuticals

US Patent
LigandPNGBDBM328072(5-(3-(4- cyanophenoxy)azetidine- 1-carbonyl)-N-(6-...)
Affinity DataEC50: >1.00E+4nMAssay Description:Compounds were assayed for their ability to activate AMPK using an enzyme-linked immunosorbent assay. Reagents and procedures for measuring AMPK acti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target5'-AMP-activated protein kinase catalytic subunit alpha-2(Homo sapiens (Human))
Rigel Pharmaceuticals

US Patent
LigandPNGBDBM328072(5-(3-(4- cyanophenoxy)azetidine- 1-carbonyl)-N-(6-...)
Affinity DataEC50: >1.00E+4nMAssay Description:Compounds were assayed for their ability to activate AMPK using an enzyme-linked immunosorbent assay. Reagents and procedures for measuring AMPK acti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent