BDBM340702 US9763922, Example 228
SMILES CC(=O)N1CCc2c(C1)c(Nc1cc(C#N)c(cc1F)-c1cn(C)nc1C(F)(F)F)nn2C1COC1
InChI Key InChIKey=KDTHDXNMPWDNBJ-UHFFFAOYSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 340702
Affinity DataIC50: 7.58E+3nMAssay Description:His/Flag epitope tagged BRD4 BD142-168 was cloned, expressed, and purified to. BRD4 binding and inhibition was assessed by monitoring the engagement ...More data for this Ligand-Target Pair
Affinity DataIC50: 82nMAssay Description:His/Flag epitope tagged CBP was cloned, expressed, and purified to homogeneity. CBP binding and inhibition was assessed by monitoring the engagement ...More data for this Ligand-Target Pair