BDBM346664 US10202379, Reference Example 263

SMILES Oc1c2C(=O)N(CC(F)(F)F)CN(C3c4ccccc4CCc4ccccc34)n2ccc1=O

InChI Key InChIKey=JRQFSJSCFALNAQ-UHFFFAOYSA-N

Data  1 IC50  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
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Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 346664   

TargetTranscription initiation factor TFIID subunit 1(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM346664(US10202379, Reference Example 263)
Affinity DataEC50:  75nMAssay Description:A test sample was diluted with a culture medium to an appropriate concentration in advance, and then 2 to 5-fold serial dilution on a 96 well plate (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTranscription initiation factor TFIID subunit 1(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM346664(US10202379, Reference Example 263)
Affinity DataIC50:  85nMAssay Description:A test sample was diluted with a culture medium to an appropriate concentration in advance, and then 2 to 5-fold serial dilution on a 96 well plate (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent