BDBM369190 3-chloro-N-[1-[6-(4-chlorophenyl)-7H- pyrrolo[2,3-d]pyrimidin-4-yl]-4- piperidyl]benzenesulfonamide::US10227357, Compound P-0480

SMILES Clc1ccc(cc1)-c1cc2c(ncnc2[nH]1)N1CCC(CC1)NS(=O)(=O)c1cccc(Cl)c1

InChI Key InChIKey=DSNINMJEUJNDDT-UHFFFAOYSA-N

Data  1 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 369190   

LigandPNGBDBM369190(US10227357, Compound P-0480 | 3-chloro-N-[1-[6-(4-...)
Affinity DataKi:  5.50E+3nMAssay Description:The c-Kit mutant D816V inhibitors were assessed using an engineered BaF3-FL KIT D816V or BaF3-FL KIT V560G/D816V cell line. The BaF3-FL KIT D816V cel...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2019
Entry Details
US Patent