BDBM369338 N-[4-[6-(2-methoxy-4-pyridyl)-7H- pyrrolo[2,3-d]pyrimidin-4-yl]cyclohex-3- en-1-yl]-4- (trifluoromethoxy)benzenesulfonamide::US10227357, Compound P-0654
SMILES COc1cc(ccn1)-c1cc2c(ncnc2[nH]1)C1=CCC(CC1)NS(=O)(=O)c1ccc(OC(F)(F)F)cc1
InChI Key
Data 2 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 369338
Affinity DataKi: 500nMAssay Description:The c-Kit mutant D816V inhibitors were assessed using an engineered BaF3-FL KIT D816V or BaF3-FL KIT V560G/D816V cell line. The BaF3-FL KIT D816V cel...More data for this Ligand-Target Pair
Affinity DataKi: 1.05E+5nMAssay Description:The c-Kit mutant D816V inhibitors were assessed using an engineered BaF3-FL KIT D816V or BaF3-FL KIT V560G/D816V cell line. The BaF3-FL KIT D816V cel...More data for this Ligand-Target Pair