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BDBM374015 (R)-2,6-difluoro-3-methyl-4-((1-(1-phenylethyl)piperidin-4-yl)oxy)-N-(thiazol-4-yl)benzenesulfonamide 2,2,2-trifluoroacetate::US10246453, Example 282::US10662184, Example 282::US10815229, Example 282::US11299490, Example 282

SMILES: C[C@@H](N1CCC(CC1)Oc1cc(F)c(c(F)c1C)S(=O)(=O)Nc1cscn1)c1ccccc1

InChI Key: InChIKey=JHYAUINCWJPVDP-UHFFFAOYSA-N

Data: 10 IC50

Find this compound or compounds like it in BindingDB or PDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 10 hits for monomerid = 374015   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kcal/mole
IC50
nM
Kd
nM
EC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Sodium channel protein type 8 subunit alpha


(Human)
BDBM374015
PNG
(US10246453, Example 282 | (R)-2,6-difluoro-3-methy...)
GoogleScholar
UniChem
n/an/a 5n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Sodium channel protein type 5 subunit alpha


(Human)
BDBM374015
PNG
(US10246453, Example 282 | (R)-2,6-difluoro-3-methy...)
GoogleScholar
UniChem
n/an/a 2.39E+4n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Sodium channel protein type 1 subunit alpha


(Human)
BDBM374015
PNG
(US10246453, Example 282 | (R)-2,6-difluoro-3-methy...)
GoogleScholar
UniChem
n/an/a 1.73E+4n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Sodium channel protein type 8 subunit alpha


(Human)
BDBM374015
PNG
(US10246453, Example 282 | (R)-2,6-difluoro-3-methy...)
GoogleScholar
UniChem
n/an/a 5n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Sodium channel protein type 8 subunit alpha


(Human)
BDBM374015
PNG
(US10246453, Example 282 | (R)-2,6-difluoro-3-methy...)
GoogleScholar
UniChem
n/an/a 5n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Sodium channel protein type 8 subunit alpha


(Human)
BDBM374015
PNG
(US10246453, Example 282 | (R)-2,6-difluoro-3-methy...)
GoogleScholar
UniChem
n/an/a 5n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Sodium channel protein type 5 subunit alpha


(Human)
BDBM374015
PNG
(US10246453, Example 282 | (R)-2,6-difluoro-3-methy...)
GoogleScholar
UniChem
n/an/a 2.39E+4n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Sodium channel protein type 1 subunit alpha


(Human)
BDBM374015
PNG
(US10246453, Example 282 | (R)-2,6-difluoro-3-methy...)
GoogleScholar
UniChem
n/an/a 1.73E+4n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Sodium channel protein type 8 subunit alpha


(Human)
BDBM374015
PNG
(US10246453, Example 282 | (R)-2,6-difluoro-3-methy...)
GoogleScholar
UniChem
n/an/a 5n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Sodium channel protein type 8 subunit alpha


(Human)
BDBM374015
PNG
(US10246453, Example 282 | (R)-2,6-difluoro-3-methy...)
GoogleScholar
UniChem
n/an/a 5n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair