BDBM378802 N-(1-((1-(4-chlorobenzyl)-1H-pyrazol-4-yl)methyl)azetidin-3-yl)-1-cyclopropyl-1H-1,2,3-triazole-4-carboxamide::US10266526, Compound 985

SMILES: c1cc(ccc1Cn2cc(cn2)CN3CC(C3)NC(=O)c4cn(nn4)C5CC5)Cl

InChI Key: InChIKey=MOWCUCXGYVJUHU-UHFFFAOYSA-N

Data: 3 IC50

PDB links: 1 PDB ID matches this monomer.

Find this compound or compounds like it in BindingDB or PDB:

Substructure Similarity at least:  must be >=0.5 Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 19 hits for monomerid = 378802   

Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50 nM	koff s-1	kon M-1s-1	pH	Temp °C
Histone-lysine N-methyltransferase PRDM9 (Homo sapiens)	BDBM378802 (US10266526, Compound 985 | N-(1-((1-(4-chlorobenzy...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
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N-lysine methyltransferase SMYD2 (Human)	BDBM378802 (US10266526, Compound 985 | N-(1-((1-(4-chlorobenzy...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	3	n/a	n/a	n/a	n/a	n/a	n/a
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Histone-lysine N-methyltransferase NSD2 (Human)	BDBM378802 (US10266526, Compound 985 | N-(1-((1-(4-chlorobenzy...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
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Histone-lysine N-methyltransferase SUV39H1 (Human)	BDBM378802 (US10266526, Compound 985 | N-(1-((1-(4-chlorobenzy...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
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Histone-lysine N-methyltransferase SETD7 (Human)	BDBM378802 (US10266526, Compound 985 | N-(1-((1-(4-chlorobenzy...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
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Histone-lysine N-methyltransferase SETD2 (Human)	BDBM378802 (US10266526, Compound 985 | N-(1-((1-(4-chlorobenzy...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
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Protein arginine N-methyltransferase 8 (Human)	BDBM378802 (US10266526, Compound 985 | N-(1-((1-(4-chlorobenzy...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
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Protein arginine N-methyltransferase 7 (Human)	BDBM378802 (US10266526, Compound 985 | N-(1-((1-(4-chlorobenzy...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
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Protein arginine N-methyltransferase 6 (Human)	BDBM378802 (US10266526, Compound 985 | N-(1-((1-(4-chlorobenzy...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
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Protein arginine N-methyltransferase 3 (Human)	BDBM378802 (US10266526, Compound 985 | N-(1-((1-(4-chlorobenzy...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
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N-lysine methyltransferase SMYD2 (Human)	BDBM378802 (US10266526, Compound 985 | N-(1-((1-(4-chlorobenzy...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	3.90	n/a	n/a	n/a	n/a	n/a	n/a
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Histone-lysine N-methyltransferase, H3 lysine-36 specific (Human)	BDBM378802 (US10266526, Compound 985 | N-(1-((1-(4-chlorobenzy...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
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Histone-lysine N-methyltransferase EZH2 (Human)	BDBM378802 (US10266526, Compound 985 | N-(1-((1-(4-chlorobenzy...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
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Histone-lysine N-methyltransferase EZH1 (Human)	BDBM378802 (US10266526, Compound 985 | N-(1-((1-(4-chlorobenzy...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
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Histone-lysine N-methyltransferase EHMT2 (Human)	BDBM378802 (US10266526, Compound 985 | N-(1-((1-(4-chlorobenzy...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
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Histone-lysine N-methyltransferase EHMT1 (Human)	BDBM378802 (US10266526, Compound 985 | N-(1-((1-(4-chlorobenzy...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
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					More data for this Ligand-Target Pair
N-lysine methyltransferase SMYD2 (Human)	BDBM378802 (US10266526, Compound 985 | N-(1-((1-(4-chlorobenzy...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	3.90	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
N-lysine methyltransferase SMYD2 (Human)	BDBM378802 (US10266526, Compound 985 | N-(1-((1-(4-chlorobenzy...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	2.90	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair
N-lysine methyltransferase SMYD2 (Human)	BDBM378802 (US10266526, Compound 985 | N-(1-((1-(4-chlorobenzy...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	3.90	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair