BDBM434905 4'-(1-(2-benzylpiperidine-1- carbonyl)-1H-1,2,3-triazol-4-yl)- 2,6-dimethoxy-N-methyl-[1,1'- biphenyl]-4-carboxamide::US10583137, Compound 79

SMILES CNC(=O)c1cc(OC)c(c(OC)c1)-c1ccc(cc1)-c1cn(nn1)C(=O)N1CCCCC1Cc1ccccc1

InChI Key InChIKey=SBLSPKKJWHIJTQ-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 434905   

TargetDiacylglycerol lipase-alpha(Human)
The Scripps Research Institute

US Patent
LigandPNGBDBM434905(US10583137, Compound 79 | 4'-(1-(2-benzylpiperidin...)
Affinity DataIC50: 1.20E+3nMAssay Description:Briefly, membrane proteome (1 mg/ml, 20 μL) was prepared from HEK293T cells (transiently transfected with hDAGLα-FLAG or hDAGLα-S472A-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2020
Entry Details
US Patent

TargetDiacylglycerol lipase-beta(Human)
The Scripps Research Institute

US Patent
LigandPNGBDBM434905(US10583137, Compound 79 | 4'-(1-(2-benzylpiperidin...)
Affinity DataIC50: 1.00E+4nMAssay Description:Briefly, membrane proteome (1 mg/ml, 20 μL) was prepared from HEK293T cells (transiently transfected with hDAGLα-FLAG or hDAGLα-S472A-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2020
Entry Details
US Patent