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BDBM4675 4-Anilinoquinazoline 22::N-(4-Bromo-2-fluorophenyl)-6-methoxy-7-(piperidin-4-ylmethoxy)quinazolin-4-amine

SMILES: COc1cc2c(Nc3ccc(Br)cc3F)ncnc2cc1OCC1CCNCC1

InChI Key: InChIKey=HTCPERSEGREUFC-UHFFFAOYSA-N

Data: 4 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 4675
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Vascular endothelial growth factor receptor 1 (Human)	BDBM4675 (N-(4-Bromo-2-fluorophenyl)-6-methoxy-7-(piperidin-...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	900	n/a	n/a	n/a	n/a	n/a	25
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Vascular endothelial growth factor receptor 2 (Human)	BDBM4675 (N-(4-Bromo-2-fluorophenyl)-6-methoxy-7-(piperidin-...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	70	n/a	n/a	n/a	n/a	n/a	25
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Fibroblast growth factor receptor 1 (Human)	BDBM4675 (N-(4-Bromo-2-fluorophenyl)-6-methoxy-7-(piperidin-...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	6.00E+3	n/a	n/a	n/a	n/a	n/a	25
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Epidermal growth factor receptor (Human)	BDBM4675 (N-(4-Bromo-2-fluorophenyl)-6-methoxy-7-(piperidin-...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	200	n/a	n/a	n/a	n/a	n/a	25
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair