BDBM469658 N-(1,1-Dimethylpropyl)-3[[2-(2-hydroxyphenyl)acetyl]amino]benzamide::US11364246, Example 1.1::US20200361871A1, Example 1.1

SMILES CN(CC1CCOC1)[C@]1(CC[C@]2(CN(C(=O)N2)c2cnc(nc2)C(F)(F)F)CC1)c1ccccc1

InChI Key InChIKey=MEKPLZGVNVGOOQ-OIPYLKGRSA-N

Data  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 469658   

TargetAnoctamin-1(Homo sapiens (Human))
Tmem16A

US Patent
LigandPNGBDBM469658(N-(1,1-Dimethylpropyl)-3[[2-(2-hydroxyphenyl)acety...)
Affinity DataEC50:  560nMAssay Description:Cell Culture and PreparationFisher rat thyroid (FRT) cells stably expressing human TMEM16A (TMEM16Aabc variant; Dr Luis Galietta, Insituto Giannina, ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAnoctamin-1(Homo sapiens (Human))
Tmem16A

US Patent
LigandPNGBDBM469658(N-(1,1-Dimethylpropyl)-3[[2-(2-hydroxyphenyl)acety...)
Affinity DataEC50:  560nMAssay Description:Compound activity was quantified by measuring the increase in current upon compound addition and expressing this as a percentage increase of baseline...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent