BDBM47125 US8952027, 63

SMILES NC(=O)c1ccc(cn1)-c1cccnc1O[C@@H]1C[C@@H](C1)Nc1ccc2ccccc2n1

InChI Key InChIKey=UPQIKAIFCRQKSJ-HDICACEKSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 47125   

TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Homo sapiens (Human))
Amgen

US Patent
LigandPNGBDBM47125(US8952027, 63)
Affinity DataIC50:  0.260nMT: 2°CAssay Description:Enzyme Activity. An IMAP TR-FRET assay was used to analyze the enzyme activity (Molecular Devices Corp., Sunnyvale Calif.). 5 uL, of serial diluted P...More data for this Ligand-Target Pair
In DepthDetails US Patent