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BDBM481128 US10906896, Cpd 809::US11725005, Compound 809

SMILES: CN1CCN(Cc2ccc(cc2)C(=O)Nc2ccc(C)c(Nc3nccc(n3)-c3cncc(c3)-c3oncc3C)c2)CC1

InChI Key: InChIKey=ADGOPPKEIZXKAZ-UHFFFAOYSA-N

Data: 1 KI 5 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 6 hits for monomerid = 481128
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Tyrosine-protein kinase ABL1 (Human)	BDBM481128 (US10906896, Cpd 809 \| US11725005, Compound 809) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	47	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Tyrosine-protein kinase ABL2 (Human)	BDBM481128 (US10906896, Cpd 809 \| US11725005, Compound 809) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	77	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Tyrosine-protein kinase ABL1 (Human)	BDBM481128 (US10906896, Cpd 809 \| US11725005, Compound 809) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	47	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Tyrosine-protein kinase ABL2 (Human)	BDBM481128 (US10906896, Cpd 809 \| US11725005, Compound 809) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	77	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Mast/stem cell growth factor receptor Kit (Human)	BDBM481128 (US10906896, Cpd 809 \| US11725005, Compound 809) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	7.80	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Mast/stem cell growth factor receptor Kit (Human)	BDBM481128 (US10906896, Cpd 809 \| US11725005, Compound 809) Show SMILES Show InChI	GoogleScholar	UniChem		7.80	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair