BDBM4852 (4-Chlorophenyl)methyl[4-(4-pyridylmethyl)phthalazin-1-yl]amine::CGP79787 Analog 37::N-(4-chlorophenyl)-N-methyl-4-(pyridin-4-ylmethyl)phthalazin-1-amine

SMILES CN(c1ccc(Cl)cc1)c1nnc(Cc2ccncc2)c2ccccc12

InChI Key InChIKey=OZGCCTRTFRHDJM-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 4852   

TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Novartis Pharmaceuticals

LigandPNGBDBM4852((4-Chlorophenyl)methyl[4-(4-pyridylmethyl)phthalaz...)
Affinity DataIC50:  3.50E+3nMAssay Description:The in vitro kinase assays were performed in 96-well plates using the recombinant GST-fused kinase domains expressed in baculovirus and purified over...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 1(Homo sapiens (Human))
Novartis Pharmaceuticals

LigandPNGBDBM4852((4-Chlorophenyl)methyl[4-(4-pyridylmethyl)phthalaz...)
Affinity DataIC50:  2.30E+3nMpH: 7.5 T: 2°CAssay Description:The in vitro kinase assays were performed in 96-well plates using the recombinant GST-fused kinase domains expressed in baculovirus and purified over...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed