Found 36 hits for monomerid = 50003659 Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
P2X purinoceptor 4
(Human) | BDBM50003659
 (5H-dibenzo[b,f]azepine-5-carboxamide | TEGRETOL | ...) | GoogleScholar
| UniChem
| | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
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Citation and Details
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More data for this Ligand-Target Pair | |
Sodium channel protein type 1/2/3 subunit alpha
(Rat) | BDBM50003659
 (5H-dibenzo[b,f]azepine-5-carboxamide | TEGRETOL | ...) | GoogleScholar
| UniChem
| | n/a | n/a | 1.31E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
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More data for this Ligand-Target Pair | |
Frizzled-8
(Mouse) | BDBM50003659
 (5H-dibenzo[b,f]azepine-5-carboxamide | TEGRETOL | ...) | GoogleScholar
| UniChem
| | n/a | n/a | n/a | 1.68E+4 | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
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More data for this Ligand-Target Pair | |
Sodium channel protein type 1 subunit alpha
(Human) | BDBM50003659
 (5H-dibenzo[b,f]azepine-5-carboxamide | TEGRETOL | ...) | GoogleScholar
| UniChem
| | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
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Citation and Details
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More data for this Ligand-Target Pair | |
Sodium channel protein type 5 subunit alpha
(Human) | BDBM50003659
 (5H-dibenzo[b,f]azepine-5-carboxamide | TEGRETOL | ...) | GoogleScholar
| UniChem
| | n/a | n/a | 4.68E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
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Citation and Details
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More data for this Ligand-Target Pair | |
Sodium channel protein type 9 subunit alpha
(Human) | BDBM50003659
 (5H-dibenzo[b,f]azepine-5-carboxamide | TEGRETOL | ...) | GoogleScholar
| UniChem
| | n/a | n/a | 9.13E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
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Citation and Details
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More data for this Ligand-Target Pair | |
Major prion protein
(Human) | BDBM50003659
 (5H-dibenzo[b,f]azepine-5-carboxamide | TEGRETOL | ...) | GoogleScholar
| UniChem
| | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
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More data for this Ligand-Target Pair | |
Sodium channel protein type 9 subunit alpha
(Human) | BDBM50003659
 (5H-dibenzo[b,f]azepine-5-carboxamide | TEGRETOL | ...) | GoogleScholar
| UniChem
| | n/a | n/a | 2.20E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
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More data for this Ligand-Target Pair | |
Potassium voltage-gated channel subfamily H member 2
(Human) | BDBM50003659
 (5H-dibenzo[b,f]azepine-5-carboxamide | TEGRETOL | ...) | GoogleScholar
| UniChem
| | n/a | n/a | 1.05E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
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More data for this Ligand-Target Pair | |
Cytochrome P450 2B6
(Human) | BDBM50003659
 (5H-dibenzo[b,f]azepine-5-carboxamide | TEGRETOL | ...) | GoogleScholar
| UniChem
| | n/a | n/a | n/a | n/a | 1.45E+5 | n/a | n/a | n/a | n/a |
TBA
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Citation and Details
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More data for this Ligand-Target Pair | |
Bile salt export pump
(Rat) | BDBM50003659
 (5H-dibenzo[b,f]azepine-5-carboxamide | TEGRETOL | ...) | GoogleScholar
| UniChem
| | n/a | n/a | >1.00E+6 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
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More data for this Ligand-Target Pair | |
Bile salt export pump
(Human) | BDBM50003659
 (5H-dibenzo[b,f]azepine-5-carboxamide | TEGRETOL | ...) | GoogleScholar
| UniChem
| | n/a | n/a | >1.00E+6 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
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Citation and Details
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More data for this Ligand-Target Pair | |
Cytochrome P450 2J2
(Human) | BDBM50003659
 (5H-dibenzo[b,f]azepine-5-carboxamide | TEGRETOL | ...) | GoogleScholar
| UniChem
| | n/a | n/a | >5.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
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Citation and Details
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More data for this Ligand-Target Pair | |
Albumin
(Rat) | BDBM50003659
 (5H-dibenzo[b,f]azepine-5-carboxamide | TEGRETOL | ...) | GoogleScholar
| UniChem
| | n/a | n/a | n/a | 1.03E+5 | n/a | n/a | n/a | n/a | n/a |
TBA
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Citation and Details
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More data for this Ligand-Target Pair | |
Sodium channel protein type 1/2/3 subunit alpha
(Rat) | BDBM50003659
 (5H-dibenzo[b,f]azepine-5-carboxamide | TEGRETOL | ...) | GoogleScholar
| UniChem
| | n/a | n/a | 1.67E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
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More data for this Ligand-Target Pair | |
Sodium channel protein type 1/2/3 subunit alpha
(Rat) | BDBM50003659
 (5H-dibenzo[b,f]azepine-5-carboxamide | TEGRETOL | ...) | GoogleScholar
| UniChem
| | n/a | n/a | 1.31E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
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More data for this Ligand-Target Pair | |
Sodium channel protein type 1/2/3 subunit alpha
(Rat) | BDBM50003659
 (5H-dibenzo[b,f]azepine-5-carboxamide | TEGRETOL | ...) | GoogleScholar
| UniChem
| | n/a | n/a | 1.31E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
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More data for this Ligand-Target Pair | |
Sodium channel protein type 1/2/3 subunit alpha
(Rat) | BDBM50003659
 (5H-dibenzo[b,f]azepine-5-carboxamide | TEGRETOL | ...) | GoogleScholar
| UniChem
| | n/a | n/a | 2.10E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
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More data for this Ligand-Target Pair | |
Sodium channel protein type 1/2/3 subunit alpha
(Rat) | BDBM50003659
 (5H-dibenzo[b,f]azepine-5-carboxamide | TEGRETOL | ...) | GoogleScholar
| UniChem
| | n/a | n/a | 1.31E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
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More data for this Ligand-Target Pair | |
ATP-binding cassette sub-family C member 2
(Human) | BDBM50003659
 (5H-dibenzo[b,f]azepine-5-carboxamide | TEGRETOL | ...) | GoogleScholar
| UniChem
| | n/a | n/a | >1.33E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
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More data for this Ligand-Target Pair | |
ATP-binding cassette sub-family C member 3
(Human) | BDBM50003659
 (5H-dibenzo[b,f]azepine-5-carboxamide | TEGRETOL | ...) | GoogleScholar
| UniChem
| | n/a | n/a | >1.33E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
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More data for this Ligand-Target Pair | |
ATP-binding cassette sub-family C member 4
(Human) | BDBM50003659
 (5H-dibenzo[b,f]azepine-5-carboxamide | TEGRETOL | ...) | GoogleScholar
| UniChem
| | n/a | n/a | >1.33E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
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More data for this Ligand-Target Pair | |
Bile salt export pump
(Human) | BDBM50003659
 (5H-dibenzo[b,f]azepine-5-carboxamide | TEGRETOL | ...) | GoogleScholar
| UniChem
| | n/a | n/a | >1.33E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
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More data for this Ligand-Target Pair | |
Bile salt export pump
(Human) | BDBM50003659
 (5H-dibenzo[b,f]azepine-5-carboxamide | TEGRETOL | ...) | GoogleScholar
| UniChem
| | n/a | n/a | >1.00E+6 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
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More data for this Ligand-Target Pair | |
Cytochrome P450 3A4
(Human) | BDBM50003659
 (5H-dibenzo[b,f]azepine-5-carboxamide | TEGRETOL | ...) | GoogleScholar
| UniChem
| | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
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More data for this Ligand-Target Pair | |
Cytochrome P450 3A4
(Human) | BDBM50003659
 (5H-dibenzo[b,f]azepine-5-carboxamide | TEGRETOL | ...) | GoogleScholar
| UniChem
| | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
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More data for this Ligand-Target Pair | |
5-hydroxytryptamine receptor 1A
(Human) | BDBM50003659
 (5H-dibenzo[b,f]azepine-5-carboxamide | TEGRETOL | ...) | GoogleScholar
| UniChem
| | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
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More data for this Ligand-Target Pair | |
5-hydroxytryptamine receptor 2A
(Rat) | BDBM50003659
 (5H-dibenzo[b,f]azepine-5-carboxamide | TEGRETOL | ...) | GoogleScholar
| UniChem
| | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
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More data for this Ligand-Target Pair | |
5-hydroxytryptamine receptor 2C
(Rat) | BDBM50003659
 (5H-dibenzo[b,f]azepine-5-carboxamide | TEGRETOL | ...) | GoogleScholar
| UniChem
| | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
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More data for this Ligand-Target Pair | |
5-hydroxytryptamine receptor 3A
(Mouse) | BDBM50003659
 (5H-dibenzo[b,f]azepine-5-carboxamide | TEGRETOL | ...) | GoogleScholar
| UniChem
| | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
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More data for this Ligand-Target Pair | |
D(1A) dopamine receptor
(Human) | BDBM50003659
 (5H-dibenzo[b,f]azepine-5-carboxamide | TEGRETOL | ...) | GoogleScholar
| UniChem
| | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
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Citation and Details
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More data for this Ligand-Target Pair | |
D(2) dopamine receptor
(Human) | BDBM50003659
 (5H-dibenzo[b,f]azepine-5-carboxamide | TEGRETOL | ...) | GoogleScholar
| UniChem
| | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
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Citation and Details
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More data for this Ligand-Target Pair | |
Glutamate receptor ionotropic, NMDA 1
(Rat) | BDBM50003659
 (5H-dibenzo[b,f]azepine-5-carboxamide | TEGRETOL | ...) | GoogleScholar
| UniChem
| | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
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More data for this Ligand-Target Pair | |
Histamine H1 receptor
(Human) | BDBM50003659
 (5H-dibenzo[b,f]azepine-5-carboxamide | TEGRETOL | ...) | GoogleScholar
| UniChem
| | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
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More data for this Ligand-Target Pair | |
Sodium channel protein type 9 subunit alpha
(Human) | BDBM50003659
 (5H-dibenzo[b,f]azepine-5-carboxamide | TEGRETOL | ...) | GoogleScholar
| UniChem
| | 3.27E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
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Citation and Details
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More data for this Ligand-Target Pair | |
Sodium channel protein type 4 subunit alpha
(Human) | BDBM50003659
 (5H-dibenzo[b,f]azepine-5-carboxamide | TEGRETOL | ...) | GoogleScholar
| UniChem
| | 5.20E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
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Citation and Details
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More data for this Ligand-Target Pair | |