BindingDB PrimarySearch

BDBM50004822 (R)-1-phenyl-2,3,4,5-tetrahydro-1H-benzo[d]azepine-7,8-diol::(R)-7,8-Dihydroxy-1-phenyl-2,3,4,5-tetrahydro-1H-benzo[d]azepinium::1-Phenyl-2,3,4,5-tetrahydro-1H-benzo[d]azepine-7,8-diol::1-Phenyl-2,3,4,5-tetrahydro-1H-benzo[d]azepine-7,8-diol(SKF38393)::7,8-Dihydroxy-1-phenyl-2,3,4,5-tetrahydro-1H-benzo[d]azepinium(R(+)SKF38393)::CHEMBL1467585::CHEMBL24077::R(+)SKF 383931-Phenyl-2,3,4,5-tetrahydro-1H-benzo[d]azepine-7,8-diol::SK&F-383933::SK-38393::SK-383933::SKF 38393::SKF 38393 (+)

SMILES: Oc1cc2CCNC[C@H](c3ccccc3)c2cc1O

InChI Key: InChIKey=JUDKOGFHZYMDMF-UHFFFAOYSA-N

Data: 46 KI 5 IC50 2 Kd 12 EC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 65 hits for monomerid = 50004822
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Adenylate cyclase type 1 (Rat)	BDBM50004822 (CHEMBL24077 \| SKF 38393 (+) \| SK-383933 \| R(+)SKF ...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	n/a	n/a	32	n/a	n/a	n/a	n/a
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D(1A) dopamine receptor (Rat)	BDBM50004822 (CHEMBL24077 \| SKF 38393 (+) \| SK-383933 \| R(+)SKF ...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	50	n/a	n/a	n/a	n/a	n/a	n/a
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D(2) dopamine receptor (Rat)	BDBM50004822 (CHEMBL24077 \| SKF 38393 (+) \| SK-383933 \| R(+)SKF ...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
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D(2) dopamine receptor (Rat)	BDBM50004822 (CHEMBL24077 \| SKF 38393 (+) \| SK-383933 \| R(+)SKF ...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a
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D(1A) dopamine receptor (Human)	BDBM50004822 (CHEMBL24077 \| SKF 38393 (+) \| SK-383933 \| R(+)SKF ...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	n/a	n/a	386	n/a	n/a	n/a	n/a
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D(1A) dopamine receptor (Rat)	BDBM50004822 (CHEMBL24077 \| SKF 38393 (+) \| SK-383933 \| R(+)SKF ...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	n/a	n/a	100	n/a	n/a	n/a	n/a
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D(1A) dopamine receptor (Human)	BDBM50004822 (CHEMBL24077 \| SKF 38393 (+) \| SK-383933 \| R(+)SKF ...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	n/a	n/a	56	n/a	n/a	n/a	n/a
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D(1A) dopamine receptor (Rat)	BDBM50004822 (CHEMBL24077 \| SKF 38393 (+) \| SK-383933 \| R(+)SKF ...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	35	n/a	n/a	n/a	n/a	n/a	n/a
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D(2) dopamine receptor (Rat)	BDBM50004822 (CHEMBL24077 \| SKF 38393 (+) \| SK-383933 \| R(+)SKF ...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	3.75E+3	n/a	n/a	n/a	n/a	n/a	n/a
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Adenylate cyclase type 5 (Human)	BDBM50004822 (CHEMBL24077 \| SKF 38393 (+) \| SK-383933 \| R(+)SKF ...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	n/a	n/a	80	n/a	n/a	n/a	n/a
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Adenylate cyclase type 1/2/3/4/5/6/7/8/9 (Human)	BDBM50004822 (CHEMBL24077 \| SKF 38393 (+) \| SK-383933 \| R(+)SKF ...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	n/a	n/a	71	n/a	n/a	n/a	n/a
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D(2) dopamine receptor (Human)	BDBM50004822 (CHEMBL24077 \| SKF 38393 (+) \| SK-383933 \| R(+)SKF ...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	n/a	n/a	>5.00E+3	n/a	n/a	n/a	n/a
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D(1A) dopamine receptor (Human)	BDBM50004822 (CHEMBL24077 \| SKF 38393 (+) \| SK-383933 \| R(+)SKF ...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	n/a	n/a	59	n/a	n/a	n/a	n/a
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D(1A)/D(1B)/D(2)/D(3)/D(4) dopamine receptor (Rat)	BDBM50004822 (CHEMBL24077 \| SKF 38393 (+) \| SK-383933 \| R(+)SKF ...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	3.39E+4	n/a	n/a	n/a	n/a	n/a	n/a
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D(2) dopamine receptor (Human)	BDBM50004822 (CHEMBL24077 \| SKF 38393 (+) \| SK-383933 \| R(+)SKF ...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a
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D(1A) dopamine receptor (Human)	BDBM50004822 (CHEMBL24077 \| SKF 38393 (+) \| SK-383933 \| R(+)SKF ...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	n/a	n/a	30	n/a	n/a	n/a	n/a
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D(2) dopamine receptor (Human)	BDBM50004822 (CHEMBL24077 \| SKF 38393 (+) \| SK-383933 \| R(+)SKF ...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	n/a	9.50E+3	n/a	n/a	n/a	n/a	n/a
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D(1) dopamine receptor (Goldfish)	BDBM50004822 (CHEMBL24077 \| SKF 38393 (+) \| SK-383933 \| R(+)SKF ...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	n/a	n/a	950	n/a	n/a	n/a	n/a
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D(1A) dopamine receptor (Human)	BDBM50004822 (CHEMBL24077 \| SKF 38393 (+) \| SK-383933 \| R(+)SKF ...) Show SMILES Show InChI	GoogleScholar	UniChem	n/a	n/a	n/a	150	n/a	n/a	n/a	n/a	n/a
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D(1A) dopamine receptor (Rat)	BDBM50004822 (CHEMBL24077 \| SKF 38393 (+) \| SK-383933 \| R(+)SKF ...) Show SMILES Show InChI	GoogleScholar	UniChem	0.300	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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D(1B) dopamine receptor (Human)	BDBM50004822 (CHEMBL24077 \| SKF 38393 (+) \| SK-383933 \| R(+)SKF ...) Show SMILES Show InChI	GoogleScholar	UniChem	0.5	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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D(1A) dopamine receptor (Human)	BDBM50004822 (CHEMBL24077 \| SKF 38393 (+) \| SK-383933 \| R(+)SKF ...) Show SMILES Show InChI	GoogleScholar	UniChem	1	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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D(1A) dopamine receptor (Human)	BDBM50004822 (CHEMBL24077 \| SKF 38393 (+) \| SK-383933 \| R(+)SKF ...) Show SMILES Show InChI	GoogleScholar	UniChem	5.10	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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D(1A) dopamine receptor (Mouse)	BDBM50004822 (CHEMBL24077 \| SKF 38393 (+) \| SK-383933 \| R(+)SKF ...) Show SMILES Show InChI	GoogleScholar	UniChem	18	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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D(1A) dopamine receptor (Rat)	BDBM50004822 (CHEMBL24077 \| SKF 38393 (+) \| SK-383933 \| R(+)SKF ...) Show SMILES Show InChI	GoogleScholar	UniChem	18	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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D(1A) dopamine receptor (Rat)	BDBM50004822 (CHEMBL24077 \| SKF 38393 (+) \| SK-383933 \| R(+)SKF ...) Show SMILES Show InChI	GoogleScholar	UniChem	18	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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D(1A) dopamine receptor (Bovine)	BDBM50004822 (CHEMBL24077 \| SKF 38393 (+) \| SK-383933 \| R(+)SKF ...) Show SMILES Show InChI	GoogleScholar	UniChem	30.4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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D(1A) dopamine receptor (Rat)	BDBM50004822 (CHEMBL24077 \| SKF 38393 (+) \| SK-383933 \| R(+)SKF ...) Show SMILES Show InChI	GoogleScholar	UniChem	35	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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D(1A) dopamine receptor (Rat)	BDBM50004822 (CHEMBL24077 \| SKF 38393 (+) \| SK-383933 \| R(+)SKF ...) Show SMILES Show InChI	GoogleScholar	UniChem	41.4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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D(1A) dopamine receptor (Human)	BDBM50004822 (CHEMBL24077 \| SKF 38393 (+) \| SK-383933 \| R(+)SKF ...) Show SMILES Show InChI	GoogleScholar	UniChem	56	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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D(1A) dopamine receptor (Rat)	BDBM50004822 (CHEMBL24077 \| SKF 38393 (+) \| SK-383933 \| R(+)SKF ...) Show SMILES Show InChI	GoogleScholar	UniChem	64	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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D(1A) dopamine receptor (Rat)	BDBM50004822 (CHEMBL24077 \| SKF 38393 (+) \| SK-383933 \| R(+)SKF ...) Show SMILES Show InChI	GoogleScholar	UniChem	64	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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D(1A) dopamine receptor (Human)	BDBM50004822 (CHEMBL24077 \| SKF 38393 (+) \| SK-383933 \| R(+)SKF ...) Show SMILES Show InChI	GoogleScholar	UniChem	73	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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D(1B) dopamine receptor (Human)	BDBM50004822 (CHEMBL24077 \| SKF 38393 (+) \| SK-383933 \| R(+)SKF ...) Show SMILES Show InChI	GoogleScholar	UniChem	100	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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D(1B) dopamine receptor (Rat)	BDBM50004822 (CHEMBL24077 \| SKF 38393 (+) \| SK-383933 \| R(+)SKF ...) Show SMILES Show InChI	GoogleScholar	UniChem	100	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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D1 dopamine receptor (Crab-eating macaque)	BDBM50004822 (CHEMBL24077 \| SKF 38393 (+) \| SK-383933 \| R(+)SKF ...) Show SMILES Show InChI	GoogleScholar	UniChem	106	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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D(1A) dopamine receptor (Human)	BDBM50004822 (CHEMBL24077 \| SKF 38393 (+) \| SK-383933 \| R(+)SKF ...) Show SMILES Show InChI	GoogleScholar	UniChem	130	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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D(1A) dopamine receptor (Human)	BDBM50004822 (CHEMBL24077 \| SKF 38393 (+) \| SK-383933 \| R(+)SKF ...) Show SMILES Show InChI	GoogleScholar	UniChem	135	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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D(1A) dopamine receptor (Human)	BDBM50004822 (CHEMBL24077 \| SKF 38393 (+) \| SK-383933 \| R(+)SKF ...) Show SMILES Show InChI	GoogleScholar	UniChem	150	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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Dopamine receptor D4 (Dog)	BDBM50004822 (CHEMBL24077 \| SKF 38393 (+) \| SK-383933 \| R(+)SKF ...) Show SMILES Show InChI	GoogleScholar	UniChem	157	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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D(1A) dopamine receptor (Human)	BDBM50004822 (CHEMBL24077 \| SKF 38393 (+) \| SK-383933 \| R(+)SKF ...) Show SMILES Show InChI	GoogleScholar	UniChem	320	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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Adenylate cyclase type 2 (Rat)	BDBM50004822 (CHEMBL24077 \| SKF 38393 (+) \| SK-383933 \| R(+)SKF ...) Show SMILES Show InChI	GoogleScholar	UniChem	415	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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D(1A) dopamine receptor (Human)	BDBM50004822 (CHEMBL24077 \| SKF 38393 (+) \| SK-383933 \| R(+)SKF ...) Show SMILES Show InChI	GoogleScholar	UniChem	987	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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D(1A) dopamine receptor (Bovine)	BDBM50004822 (CHEMBL24077 \| SKF 38393 (+) \| SK-383933 \| R(+)SKF ...) Show SMILES Show InChI	GoogleScholar	UniChem	1.35E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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D(2) dopamine receptor (Rat)	BDBM50004822 (CHEMBL24077 \| SKF 38393 (+) \| SK-383933 \| R(+)SKF ...) Show SMILES Show InChI	GoogleScholar	UniChem	1.62E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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Dopamine receptor D4 (Dog)	BDBM50004822 (CHEMBL24077 \| SKF 38393 (+) \| SK-383933 \| R(+)SKF ...) Show SMILES Show InChI	GoogleScholar	UniChem	1.80E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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D(2) dopamine receptor (Rat)	BDBM50004822 (CHEMBL24077 \| SKF 38393 (+) \| SK-383933 \| R(+)SKF ...) Show SMILES Show InChI	GoogleScholar	UniChem	2.90E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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5-hydroxytryptamine receptor 1A (Human)	BDBM50004822 (CHEMBL24077 \| SKF 38393 (+) \| SK-383933 \| R(+)SKF ...) Show SMILES Show InChI	GoogleScholar	UniChem	3.10E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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D(2) dopamine receptor (Human)	BDBM50004822 (CHEMBL24077 \| SKF 38393 (+) \| SK-383933 \| R(+)SKF ...) Show SMILES Show InChI	GoogleScholar	UniChem	4.67E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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D(3) dopamine receptor (Rat)	BDBM50004822 (CHEMBL24077 \| SKF 38393 (+) \| SK-383933 \| R(+)SKF ...) Show SMILES Show InChI	GoogleScholar	UniChem	5.00E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
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